SCHEMBL8916514

SCHEMBL8916514

O=C1Cc2cc([S+]([O-])CCCN3CCC(c4noc5cc(F)ccc45)CC3)sc2CN1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.51
DRD2 P14416 4/20 0.51
SLC6A4 P31645 1/20 0.51
HTR2A P28223 2/20 0.51
HTR2C P28335 5/20 0.49
HTR6 P50406 2/20 0.48
HTR1A P08908 1/20 0.48
ADRA1A P35348 1/20 0.48
HRH1 P35367 1/20 0.48
DRD3 P35462 1/20 0.48
KCNH2 Q12809 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8917771 0.84 DRD2 (0.58) ACHEDRD2SLC6A4HTR2AHTR2C
SCHEMBL8918416 0.84 HTR2A (0.53) ACHEDRD2SLC6A4HTR2AHTR2C
SCHEMBL8917294 0.84 ACHE (0.52) ACHEDRD2SLC6A4HTR2AHTR2C
SCHEMBL8920261 0.84 DRD2 (0.58) ACHEDRD2SLC6A4HTR2AHTR2C
SCHEMBL8920476 0.84 ACHE (0.52) ACHEDRD2SLC6A4HTR2AHTR2C
SCHEMBL8917083 0.80 ACHE (0.50) ACHEDRD2SLC6A4HTR2AHTR2C
SCHEMBL8917276 0.78 HTR2C (0.58) ACHEDRD2SLC6A4HTR2AHTR2C
Oxalic Acid SCHEMBL9141181 0.74 HTR2A (0.60) DRD2SLC6A4HTR2AHTR2CHTR6
SCHEMBL8918221 0.73 ACHE (0.50) ACHEDRD2SLC6A4HTR2AHTR2C
SCHEMBL1545611 0.73 ACHE (0.93) ACHEDRD2SLC6A4HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691330-A ANTIPSYCHOTIC AGENT YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-11-25 US disclosed
US-5532240-A ANTIPSYCHOTIC AGENTS AND ANTISEROTONIN AGENTS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-07-02 US disclosed
EP-0596125-A1 CONDENSED THIOPHENE COMPOUND AND PHARMACEUTICAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1994-05-11 EP disclosed