SCHEMBL8916684

SCHEMBL8916684

NC(=O)c1ccc2c(OC(=O)c3ccccc3C(=O)Oc3c[nH]c4cc(C(N)=O)ccc34)c[nH]c2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A6 Q4U2R8 1/20 0.44
ALDH1A1 P00352 1/20 0.41
ATM Q13315 1/20 0.41
ASH1L Q9NR48 2/20 0.40
MEN1 O00255 1/20 0.40
CYP1A2 P05177 1/20 0.40
HTR1A P08908 1/20 0.40
TSHR P16473 1/20 0.40
HTR1D P28221 1/20 0.40
HTR1B P28222 1/20 0.40
HTR2C P28335 1/20 0.40
HTR7 P34969 1/20 0.40
HTR5A P47898 1/20 0.40
HTR6 P50406 1/20 0.40
KMT2A Q03164 1/20 0.40
HSD17B10 Q99714 1/20 0.40
NR4A2 P43354 2/20 0.40
PARP1 P09874 2/20 0.39
PRSS1 P07477 1/20 0.39
ACR P10323 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8915831 0.89 PARP10 (0.50) SLC22A6ALDH1A1ATMASH1LMEN1
SCHEMBL8915869 0.84 HTR1B (0.44) SLC22A6ASH1LMEN1CYP1A2HTR1A
SCHEMBL8914633 0.82 SLC22A6 (0.59) SLC22A6ALDH1A1ASH1LMEN1CYP1A2
SCHEMBL8915441 0.81 HTR1D (0.45) SLC22A6ASH1LMEN1CYP1A2HTR1A
SCHEMBL8917348 0.81 PLG (0.43) SLC22A6ALDH1A1ASH1LMEN1CYP1A2
SCHEMBL8915273 0.81 HTR1A (0.45) SLC22A6ALDH1A1ASH1LMEN1CYP1A2
SCHEMBL8915816 0.81 PLG (0.43) SLC22A6ALDH1A1ASH1LMEN1CYP1A2
SCHEMBL28515587 0.79 SLC22A6 (0.68) SLC22A6ALDH1A1ATMMEN1CYP1A2
SCHEMBL8917363 0.78 KMT2A (0.43) SLC22A6ALDH1A1ASH1LMEN1CYP1A2
SCHEMBL28842060 0.78 SLC22A6 (0.41) SLC22A6ASH1LMEN1CYP1A2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5703112-A Method of preventing emesis using tetrahydrobenz CD!indole-6-carbonxamides ELI LILLY AND COMPANY (US) 1997-12-30 US disclosed