SCHEMBL8916695

SCHEMBL8916695

N#Cc1ccc(Cn2c(-c3ccccc3)c(-c3ccccc3)n(Cc3ccc4ccc(C#N)cc4c3)c2=O)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 1/20 0.49
HDAC8 Q9BY41 2/20 0.44
HDAC6 Q9UBN7 2/20 0.44
HDAC1 Q13547 1/20 0.44
CNR1 P21554 1/20 0.41
PGR P06401 3/20 0.41
CYP19A1 P11511 2/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
AR P10275 1/20 0.41
USP2 O75604 1/20 0.41
POLB P06746 1/20 0.41
TSHR P16473 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
BRD4 O60885 1/20 0.40
DRD2 P14416 1/20 0.40
TBXA2R P21731 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
PRMT5 O14744 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8440634 0.97 CFTR (0.48) CFTRHDAC8HDAC6HDAC1CNR1
SCHEMBL8908297 0.93 CFTR (0.53) CFTRHDAC8HDAC6HDAC1CNR1
SCHEMBL8441589 0.88 CFTR (0.49) CFTRHDAC8HDAC6HDAC1CNR1
SCHEMBL8908061 0.88 CFTR (0.57) CFTRHDAC8HDAC6HDAC1CNR1
SCHEMBL8439957 0.82 CFTR (0.58) CFTRHDAC8HDAC6HDAC1CNR1
SCHEMBL7359654 0.75 PRMT5 (0.57) HDAC8HDAC6HDAC1CYP19A1AR
SCHEMBL8487543 0.75 CFTR (0.54) CFTRHDAC8HDAC6CNR1AR
SCHEMBL7360668 0.74 F2 (0.54)
SCHEMBL7366139 0.73 F10 (0.53)
SCHEMBL8907770 0.73 CFTR (0.49) CFTRHDAC8HDAC6CNR1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5612363-A FACTOR XA INHIBITORS BERLEX LABORATORIES, INC. (US) 1997-03-18 US disclosed