SCHEMBL8916752

SCHEMBL8916752

NC(=O)CCN1CCC[C@@H]1Cc1c[nH]c2ccc(Br)cc12

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 5/20 0.49
HTR1B P28222 7/20 0.49
HTR1D P28221 5/20 0.49
SLC6A4 P31645 1/20 0.48
HTR1A P08908 3/20 0.47
NOS3 P29474 4/20 0.44
NOS1 P29475 4/20 0.44
UTS2R Q9UKP6 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8886632 0.87 HTR6 (0.51) HTR6HTR1BHTR1DSLC6A4HTR1A
SCHEMBL8886182 0.87 HTR6 (0.49) HTR6HTR1BHTR1DSLC6A4HTR1A
SCHEMBL8915023 0.81 HTR1B (0.51) HTR6HTR1BHTR1DHTR1ANOS3
SCHEMBL8885771 0.81 HTR1B (0.59) HTR6HTR1BHTR1DSLC6A4HTR1A
Oxalic Acid SCHEMBL2727283 0.81 HTR1B (0.68) HTR6HTR1BHTR1DHTR1A
Oxalic Acid SCHEMBL2725284 0.81 HTR1B (0.68) HTR6HTR1BHTR1DHTR1A
SCHEMBL9033153 0.81 HTR1B (0.47) HTR6HTR1BHTR1DHTR1ANOS3
SCHEMBL9033149 0.81 HTR1B (0.47) HTR6HTR1BHTR1DHTR1ANOS3
SCHEMBL8885806 0.81 SLC6A4 (0.57) HTR6HTR1BHTR1DSLC6A4HTR1A
SCHEMBL9545605 0.79 HTR1B (0.46) HTR6HTR1BHTR1DHTR1ANOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607960-A Indole derivatives as 5-HT1-like agonists for use in migraine PFIZER INC. (US) 1997-03-04 US disclosed
EP-0695301-B1 INDOLE DERIVATIVES AS 5-HT1-LIKE AGONISTS FOR USE IN MIGRAINE PFIZER LTD (GB) 1996-10-30 EP disclosed
WO-1994024127-A1 INDOLE DERIVATIVES AS 5-H1-LIKE AGONISTS FOR USE IN MIGRAINE PFIZER LIMITED (GB) 1994-10-27 WO disclosed