SCHEMBL8917374

SCHEMBL8917374

C/C=C(/C=C/CSc1ncnc2[nH]cnc12)CC

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PAK1 Q13153 1/20 0.32
TSHR P16473 1/20 0.31
NOTUM Q6P988 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8917375 0.80 PAK1 (0.54) PAK1TSHR
SCHEMBL2115552 0.76 PAK1 (0.40) PAK1TSHRNOTUM
SCHEMBL10426488 0.75 SMN1; SMN2 (0.41) PAK1TSHRNOTUM
SCHEMBL29951296 0.75 NOTUM (0.36) PAK1TSHRNOTUM
SCHEMBL2118555 0.73 PAK1 (0.48) PAK1TSHRNOTUM
SCHEMBL14028465 0.71 CYP1A2 (0.54) TSHR
SCHEMBL1725582 0.70 PAK1 (0.62) PAK1
SCHEMBL735449 0.69 NOTUM (0.60) TSHRNOTUM
SCHEMBL10927535 0.69 PAK1 (0.61) PAK1
SCHEMBL10925300 0.69 PAK1 (0.61) PAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691366-A UNSATURATED NITRO OXIME FORMED BY REACTION OF DINITROGEN TRIOXIDE WITH DIOLEFIN ETHER, SULFIDE OR AMINE TO BE USED AS VASODILATORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-11-25 US disclosed
US-5495023-A VASODILATORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-02-27 US disclosed
WO-1993010097-A1 NITRO COMPOUNDS HAVING VASODILATOR ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-05-27 WO disclosed