SCHEMBL8917375

SCHEMBL8917375

CC=C(C=CCSc1ncnc2nc[nH]c12)CC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PAK1 Q13153 1/20 0.54
TSHR P16473 1/20 0.53
MAPT P10636 1/20 0.50
HIF1A Q16665 2/20 0.49
HSD17B10 Q99714 2/20 0.49
TP53 P04637 2/20 0.49
CDC7 O00311 6/20 0.48
DBF4 Q9UBU7 6/20 0.48
G6PD P11413 1/20 0.48
LMNA P02545 5/20 0.46
HTT P42858 4/20 0.46
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
HPGD P15428 3/20 0.45
ALDH1A1 P00352 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4253200 0.80 TSHR (0.60) PAK1TSHRMAPTHIF1AHSD17B10
SCHEMBL8917374 0.80 PAK1 (0.32) PAK1TSHR
SCHEMBL2115555 0.76 PAK1 (0.71) PAK1TSHRMAPTHIF1AHSD17B10
SCHEMBL31439407 0.76 PAK1 (0.71) PAK1TSHRMAPTHIF1AHSD17B10
SCHEMBL10426489 0.75 G6PD (0.64) PAK1TSHRMAPTHIF1AHSD17B10
SCHEMBL8642694 0.70 PAK1 (0.97) PAK1TSHRMAPTHIF1AHSD17B10
SCHEMBL10927540 0.70 PAK1 (0.97) PAK1TSHRMAPTHIF1AHSD17B10
SCHEMBL3396404 0.69 TSHR (0.78) PAK1TSHRMAPTHIF1ACDC7
SCHEMBL240980 0.67 HSD17B10 (1.00) PAK1TSHRMAPTHIF1AHSD17B10
SCHEMBL30132912 0.67 HSD17B10 (1.00) PAK1TSHRMAPTHIF1AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691366-A UNSATURATED NITRO OXIME FORMED BY REACTION OF DINITROGEN TRIOXIDE WITH DIOLEFIN ETHER, SULFIDE OR AMINE TO BE USED AS VASODILATORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-11-25 US disclosed
US-5495023-A VASODILATORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-02-27 US disclosed
EP-0612315-A1 NITRO COMPOUNDS HAVING VASODILATOR ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-08-31 EP disclosed
WO-1993010097-A1 NITRO COMPOUNDS HAVING VASODILATOR ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-05-27 WO disclosed