SCHEMBL8917786

SCHEMBL8917786

NS(=O)(=O)c1ccc(-n2nc(C(F)F)c3ccc4c[c]ccc4c32)cc1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.40
PTGS1 P23219 9/20 0.40
PDPK1 O15530 4/20 0.37
CA12 O43570 2/20 0.36
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
CA9 Q16790 2/20 0.36
ABCB11 O95342 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8917487 0.89 PTGS2 (0.36) PTGS2PTGS1
SCHEMBL8917480 0.82 PTGS2 (0.49) PTGS2PTGS1PDPK1
SCHEMBL9235959 0.82 PTGS2 (0.53) PTGS2PTGS1PDPK1CA12CA1
SCHEMBL9231444 0.82 PTGS2 (0.44) PTGS2PTGS1PDPK1CA1CA2
SCHEMBL9231983 0.81 PTGS2 (0.43) PTGS2PTGS1PDPK1CA9
SCHEMBL9229656 0.81 PTGS2 (0.45) PTGS2PTGS1PDPK1CA12CA1
SCHEMBL9233935 0.81 PTGS2 (0.52) PTGS2PTGS1PDPK1
SCHEMBL9232444 0.78 PTGS2 (0.54) PTGS2PTGS1CA1CA2CA9
SCHEMBL8918143 0.78 PTGS2 (0.54) PTGS2PTGS1PDPK1CA12CA1
SCHEMBL9233583 0.72 PTGS2 (0.52) PTGS2PTGS1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5696143-A ARTHRITIS THERAPY G.D. SEARLE & CO. 1997-12-09 US disclosed