SCHEMBL8917480

SCHEMBL8917480

NS(=O)(=O)c1ccc(-n2nc(C(F)(F)F)c3ccc4c[c]ccc4c32)cc1

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.49
PTGS1 P23219 11/20 0.49
PDPK1 O15530 5/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8917478 0.89 CYP1A2 (0.47) PTGS2PTGS1
SCHEMBL9233871 0.84 PDPK1 (0.60) PTGS2PTGS1PDPK1
SCHEMBL8917786 0.82 PTGS2 (0.40) PTGS2PTGS1PDPK1
SCHEMBL7651780 0.82 PTGS2 (0.54) PTGS2PTGS1PDPK1
SCHEMBL9229049 0.81 PTGS2 (0.55) PTGS2PTGS1PDPK1
SCHEMBL8917361 0.79 PTGS2 (0.56) PTGS2PTGS1PDPK1
SCHEMBL9233734 0.78 PTGS2 (0.57) PTGS2PTGS1PDPK1
SCHEMBL8918086 0.75 PTGS2 (0.48) PTGS2PTGS1PDPK1
SCHEMBL9091738 0.75 PTGS2 (0.58) PTGS2PTGS1PDPK1
SCHEMBL7649968 0.74 PTGS2 (0.53) PTGS2PTGS1PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5696143-A ARTHRITIS THERAPY G.D. SEARLE & CO. 1997-12-09 US disclosed