SCHEMBL8918403

SCHEMBL8918403

CCC(C=CCNC(=O)c1cccnc1)=CC(C)C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.49
KMT2A Q03164 4/20 0.48
MEN1 O00255 3/20 0.48
NPC1 O15118 4/20 0.47
RAB9A P51151 4/20 0.47
SMN1; SMN2 Q16637 4/20 0.47
TP53 P04637 2/20 0.47
ALDH1A1 P00352 2/20 0.47
NPSR1 Q6W5P4 2/20 0.47
GAA P10253 3/20 0.47
HDAC3 O15379 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
ROCK2 O75116 1/20 0.45
ROCK1 Q13464 1/20 0.45
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
EPHX2 P34913 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8918397 1.00 THRB (0.49) THRBKMT2AMEN1NPC1RAB9A
SCHEMBL8921547 0.88 THRB (0.54) THRBKMT2AMEN1NPC1RAB9A
SCHEMBL8920234 0.88 THRB (0.54) THRBKMT2AMEN1NPC1RAB9A
SCHEMBL8921545 0.88 THRB (0.54) THRBKMT2AMEN1NPC1RAB9A
SCHEMBL8918589 0.81 THRB (0.54) THRBKMT2AMEN1NPC1RAB9A
SCHEMBL8918592 0.81 THRB (0.54) THRBKMT2AMEN1NPC1RAB9A
SCHEMBL8921909 0.78 THRB (0.56) THRBKMT2AMEN1NPC1RAB9A
SCHEMBL8921907 0.78 THRB (0.56) THRBKMT2AMEN1NPC1RAB9A
SCHEMBL8918394 0.77 THRB (0.52) THRBKMT2AMEN1NPC1RAB9A
SCHEMBL8919867 0.77 THRB (0.52) THRBKMT2AMEN1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691366-A UNSATURATED NITRO OXIME FORMED BY REACTION OF DINITROGEN TRIOXIDE WITH DIOLEFIN ETHER, SULFIDE OR AMINE TO BE USED AS VASODILATORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-11-25 US disclosed
US-5495023-A VASODILATORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-02-27 US disclosed
EP-0612315-A1 NITRO COMPOUNDS HAVING VASODILATOR ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-08-31 EP disclosed
WO-1993010097-A1 NITRO COMPOUNDS HAVING VASODILATOR ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-05-27 WO disclosed