SCHEMBL8921547

SCHEMBL8921547

CC=C(C=CCNC(=O)c1cccnc1)CC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.54
RAB9A P51151 5/20 0.49
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
NPC1 O15118 3/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
GAA P10253 3/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
EPHX2 P34913 1/20 0.48
SREBF2 Q12772 1/20 0.47
NPSR1 Q6W5P4 2/20 0.47
MAPT P10636 1/20 0.47
GFER P55789 1/20 0.47
HDAC1 Q13547 3/20 0.47
HDAC6 Q9UBN7 2/20 0.47
HDAC3 O15379 2/20 0.46
HDAC2 Q92769 2/20 0.46
TSHR P16473 1/20 0.46
ROCK2 O75116 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8921545 1.00 THRB (0.54) THRBRAB9AMEN1KMT2ANPC1
SCHEMBL8920234 1.00 THRB (0.54) THRBRAB9AMEN1KMT2ANPC1
SCHEMBL8918397 0.88 THRB (0.49) THRBRAB9AMEN1KMT2ANPC1
SCHEMBL8918403 0.88 THRB (0.49) THRBRAB9AMEN1KMT2ANPC1
SCHEMBL8921907 0.84 THRB (0.56) THRBRAB9AMEN1KMT2ANPC1
SCHEMBL8921909 0.84 THRB (0.56) THRBRAB9AMEN1KMT2ANPC1
SCHEMBL8919987 0.84 SMN1; SMN2 (0.55) RAB9AKMT2ASMN1; SMN2GAACYP1A2
SCHEMBL8918592 0.82 THRB (0.54) THRBRAB9AMEN1KMT2ANPC1
SCHEMBL8919032 0.82 KDM4E (0.51) RAB9AKMT2ANPC1SMN1; SMN2CYP1A2
SCHEMBL8918589 0.82 THRB (0.54) THRBRAB9AMEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691366-A UNSATURATED NITRO OXIME FORMED BY REACTION OF DINITROGEN TRIOXIDE WITH DIOLEFIN ETHER, SULFIDE OR AMINE TO BE USED AS VASODILATORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-11-25 US disclosed
US-5495023-A VASODILATORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-02-27 US disclosed
EP-0612315-A1 NITRO COMPOUNDS HAVING VASODILATOR ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-08-31 EP disclosed
WO-1993010097-A1 NITRO COMPOUNDS HAVING VASODILATOR ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-05-27 WO disclosed