SCHEMBL8918437

SCHEMBL8918437

O=C1NCCCc2cc(CCCl)sc21

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.35
CDK1 P06493 1/20 0.35
MAPKAPK2 P49137 1/20 0.35
TSHR P16473 1/20 0.33
PRKD1 Q15139 1/20 0.31
PRF1 P14222 1/20 0.31
ATM Q13315 1/20 0.30
USP2 O75604 1/20 0.30
MAPK1 P28482 1/20 0.30
HTT P42858 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24733658 0.76 CDK1 (0.39) ALDH1A1CDK1MAPKAPK2TSHRPRKD1
SCHEMBL8915748 0.74 GSK3B (0.43) ALDH1A1CDK1MAPKAPK2TSHRUSP2
SCHEMBL23142246 0.73 CDK1 (0.42) ALDH1A1CDK1MAPKAPK2TSHRPRKD1
SCHEMBL23177730 0.73 CDK1 (0.39) ALDH1A1CDK1MAPKAPK2TSHRPRKD1
SCHEMBL8916133 0.73 NOTUM (0.33) ALDH1A1CDK1MAPKAPK2TSHRPRKD1
SCHEMBL3974015 0.66 TSHR (0.38) ALDH1A1CDK1MAPKAPK2TSHRPRKD1
SCHEMBL26117612 0.66 PARP10 (0.34) ALDH1A1USP2MAPK1HTTTDP1
SCHEMBL26112293 0.65 USP2 (0.33) ALDH1A1PRKD1USP2MAPK1HTT
SCHEMBL13361329 0.63 PARP10 (0.46) CDK1MAPKAPK2TSHR
SCHEMBL390545 0.63 PARP10 (0.46) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691330-A ANTIPSYCHOTIC AGENT YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-11-25 US disclosed
US-5532240-A ANTIPSYCHOTIC AGENTS AND ANTISEROTONIN AGENTS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-07-02 US disclosed
EP-0596125-A1 CONDENSED THIOPHENE COMPOUND AND PHARMACEUTICAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1994-05-11 EP disclosed