SCHEMBL8916133

SCHEMBL8916133

O=C(CCCCl)c1cc2c(s1)C(=O)NCCC2

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.33
CDK1 P06493 1/20 0.32
MAPKAPK2 P49137 1/20 0.32
ALDH1A1 P00352 3/20 0.32
USP2 O75604 1/20 0.31
MAPK1 P28482 1/20 0.31
HTT P42858 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
NNMT P40261 1/20 0.31
GSK3B P49841 2/20 0.31
MAPK14 Q16539 1/20 0.31
KDM4E B2RXH2 1/20 0.30
MAPT P10636 1/20 0.30
TSHR P16473 1/20 0.30
PRKD1 Q15139 1/20 0.30
DAO P14920 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8915748 0.87 GSK3B (0.43) NOTUMCDK1MAPKAPK2ALDH1A1USP2
SCHEMBL8917631 0.80 CDC7 (0.35) ALDH1A1GSK3BMAPK14DAO
SCHEMBL8918437 0.73 ALDH1A1 (0.35) CDK1MAPKAPK2ALDH1A1USP2MAPK1
SCHEMBL24733658 0.70 CDK1 (0.39) CDK1MAPKAPK2ALDH1A1KDM4EMAPT
SCHEMBL8991820 0.70 RYR2 (0.33) GSK3BMAPK14PRKD1
SCHEMBL23177730 0.68 CDK1 (0.39) CDK1MAPKAPK2ALDH1A1MAPK1HTT
SCHEMBL23142246 0.68 CDK1 (0.42) CDK1MAPKAPK2ALDH1A1USP2MAPK1
SCHEMBL8918044 0.68 ALDH1A1 (0.33) ALDH1A1USP2MAPK1HTTTDP1
SCHEMBL8917854 0.66 PARP1 (0.35) ALDH1A1
SCHEMBL1393398 0.65 ALDH1A1 (0.60) ALDH1A1MAPK1HTTKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691330-A ANTIPSYCHOTIC AGENT YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-11-25 US disclosed
US-5532240-A ANTIPSYCHOTIC AGENTS AND ANTISEROTONIN AGENTS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-07-02 US disclosed
EP-0596125-A1 CONDENSED THIOPHENE COMPOUND AND PHARMACEUTICAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1994-05-11 EP disclosed