SCHEMBL8918845

SCHEMBL8918845

CS(=O)(=O)c1ccc(-c2nnsc2-c2cccc(Cl)c2)cc1

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.62
LMNA P02545 2/20 0.46
MAPT P10636 2/20 0.46
NPSR1 Q6W5P4 2/20 0.46
NFKB1 P19838 1/20 0.46
NFKB2 Q00653 1/20 0.46
KMT2A Q03164 1/20 0.46
RELA Q04206 1/20 0.46
SCD O00767 1/20 0.45
FLT3 P36888 1/20 0.43
S1PR4 O95977 1/20 0.43
S1PR1 P21453 1/20 0.43
HTT P42858 1/20 0.43
FAAH O00519 1/20 0.43
KCNH2 Q12809 1/20 0.43
PTGS1 P23219 3/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
RORC P51449 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8918839 0.95 PTGS2 (0.62) PTGS2LMNAMAPTNPSR1NFKB1
SCHEMBL8918438 0.85 PTGS2 (0.74) PTGS2LMNAMAPTKMT2ASCD
SCHEMBL8918833 0.84 PTGS2 (0.76) PTGS2LMNAMAPTNPSR1NFKB1
SCHEMBL8918835 0.84 PTGS2 (0.76) PTGS2LMNAMAPTNPSR1NFKB1
SCHEMBL8917019 0.82 PTGS2 (0.73) PTGS2PTGS1
SCHEMBL8918427 0.80 PTGS2 (0.74) PTGS2SCDPTGS1
SCHEMBL8915742 0.77 PTGS2 (0.80) PTGS2LMNAMAPTKMT2AHTT
SCHEMBL8918347 0.77 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL8918341 0.77 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL8917014 0.76 PTGS2 (0.73) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5677318-A Diphenyl-1,2-3-thiadiazoles as anti-inflammatory agents MERCK FROSST CANADA, INC. (CA) 1997-10-14 US claimed
US-5677318-A Diphenyl-1,2-3-thiadiazoles as anti-inflammatory agents MERCK FROSST CANADA, INC. (CA) 1997-10-14 US disclosed