SCHEMBL8918930

SCHEMBL8918930

N#CNC(=Nc1ccncc1)NCCCCCCSc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 13/20 0.48
HRH2 P25021 9/20 0.48
HRH1 P35367 5/20 0.47
HRH3 Q9Y5N1 5/20 0.47
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
HIF1A Q16665 1/20 0.37
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8916216 0.99 HRH4 (0.48) HRH4HRH2HRH1HRH3CYP1A2
SCHEMBL8915041 0.91 HRH4 (0.53) HRH4HRH2HRH1HRH3CYP1A2
SCHEMBL8918620 0.85 MAPT (0.45) HRH4HRH2HRH1HRH3HDAC3
SCHEMBL504459 0.83 CYP3A4 (0.47) HRH4HRH2HRH3CYP3A4CYP2D6
SCHEMBL504267 0.83 CYP3A4 (0.47) HRH4HRH2HRH3CYP3A4CYP2D6
SCHEMBL8054318 0.83 CYP3A4 (0.47) HRH4HRH2HRH3CYP3A4CYP2D6
SCHEMBL504467 0.83 CYP3A4 (0.47) HRH4HRH2HRH3CYP3A4CYP2D6
SCHEMBL504458 0.83 CYP3A4 (0.47) HRH4HRH2HRH3CYP3A4CYP2D6
SCHEMBL8054097 0.83 CYP3A4 (0.47) HRH4HRH2HRH3CYP3A4CYP2D6
SCHEMBL504466 0.83 CYP3A4 (0.47) HRH4HRH2HRH3CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5696140-A FOR TREATMENT OF ASTHMA, ALLERGIES, NERVOUS SYSTEM DISORDERS OR CANCER LEO PHARMACEUTICAL PRODUCTS LTD. (DK) 1997-12-09 US disclosed