SCHEMBL8919147

SCHEMBL8919147

CCn1c(=O)oc2cc(CBr)cnc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 1/20 0.37
PDE10A Q9Y233 2/20 0.35
PIK3CD O00329 2/20 0.33
NPC1 O15118 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PDE4B Q07343 1/20 0.32
MIF P14174 2/20 0.31
CD74 P04233 1/20 0.31
HSD17B10 Q99714 1/20 0.30
HPGD P15428 1/20 0.30
CRHBP P24387 1/20 0.30
HTT P42858 1/20 0.30
CRHR2 Q13324 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
MEN1 O00255 1/20 0.30
POLB P06746 1/20 0.30
KMT2A Q03164 1/20 0.30
PTGER4 P35408 1/20 0.30
IDO1 P14902 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8624408 0.89 ALDH1A1 (0.36) ALDH1A1KDM4EPDE10APIK3CDNPC1
SCHEMBL17418888 0.83 PDE4B (0.43) ALDH1A1KDM4EPDE10APIK3CDNPC1
SCHEMBL8624806 0.82 HSD17B10 (0.35) ALDH1A1KDM4EPDE10ASMN1; SMN2HSD17B10
SCHEMBL31667522 0.79 NPC1 (0.35) ALDH1A1KDM4ENPC1
SCHEMBL8917229 0.77 ALDH1A1 (0.36) ALDH1A1KDM4EPDE10APIK3CDSMN1; SMN2
SCHEMBL8918838 0.72 DRD4 (0.51) KMT2A
SCHEMBL17418949 0.71 GSK3A (0.37) ALDH1A1KDM4ESMN1; SMN2
SCHEMBL25865421 0.68 ALDH1A1 (0.43) ALDH1A1KDM4EPDE10APIK3CDNPC1
SCHEMBL25865370 0.67 HSD17B10 (0.45) ALDH1A1KDM4EPDE10ANPC1SMN1; SMN2
SCHEMBL7316292 0.66 NPC1 (0.63) ALDH1A1KDM4EPIK3CDNPC1MIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5618819-A ANALGESICS ADIR ET COMPAGNIE (FR) 1997-04-08 US disclosed
EP-0691339-A1 Amine derivatives of 1,3-dihydro-2H-pyrrolo(2,3-b)pyridin-2-ones and oxazolo(4,5-b)pyridin-2(3H)-ones, their process of preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-01-10 EP disclosed