SCHEMBL8919347

SCHEMBL8919347

Cc1ccc2c(c1)C(c1ccccc1)CC(Br)C(=O)N2

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 6/20 0.44
KMT2A Q03164 6/20 0.44
TP53 P04637 2/20 0.42
GAA P10253 1/20 0.41
ALDH1A1 P00352 1/20 0.41
ALDH2 P05091 1/20 0.41
ATM Q13315 1/20 0.41
CYP19A1 P11511 2/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
DDB1 Q16531 1/20 0.39
CRBN Q96SW2 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8399414 0.90 ALDH1A1 (0.44) MEN1KMT2ATP53ALDH1A1ALDH2
SCHEMBL8923872 0.84 ATM (0.45) MEN1KMT2ATP53GAAATM
SCHEMBL8920778 0.84 MAPT (0.42) MEN1KMT2AALDH1A1CYP19A1DDB1
SCHEMBL8400979 0.83 DDB1 (0.45) MEN1KMT2AALDH1A1DDB1CRBN
SCHEMBL8398575 0.81 THRB (0.42) MEN1KMT2AALDH1A1ALDH2SLC6A2
SCHEMBL8921539 0.78 DDB1 (0.55) MEN1KMT2ATP53GAAALDH1A1
SCHEMBL12559670 0.78 TDP1 (0.57) MEN1KMT2ATP53GAAALDH1A1
SCHEMBL8398580 0.76 SLC6A2 (0.43) TP53ALDH1A1CYP19A1SLC6A2SLC6A4
SCHEMBL18025749 0.76 BRD4 (0.57) MEN1KMT2ATP53GAAATM
SCHEMBL8402167 0.75 DDB1 (0.47) MEN1KMT2ATP53ALDH1A1DDB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5643904-A Substituted hexahdryoazepinones and tetrahydrobenzazepinones PFIZER INC. (US) 1997-07-01 US disclosed
US-5484917-A FOR TREATMENT AND PREVENTION OF GASTROINTESTINAL DISORDERS, PAIN AND ANXIETY PFIZER INC. (US) 1996-01-16 US disclosed