SCHEMBL8919912

SCHEMBL8919912

COc1ccccc1C([CH]Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)N1CCN(C(C)c2ccccc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 18/20 0.46
CYP2D6 P10635 1/20 0.40
AURKA O14965 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8919968 0.91 TACR1 (0.47) TACR1
SCHEMBL8671580 0.90 TACR1 (0.49) TACR1
SCHEMBL8673617 0.88 TACR1 (0.49) TACR1
SCHEMBL8672306 0.87 CYP2D6 (0.48) TACR1CYP2D6
SCHEMBL8673323 0.87 TACR1 (0.47) TACR1
SCHEMBL8924107 0.86 TACR1 (0.46) TACR1
SCHEMBL8676401 0.84 KCNH2 (0.47) TACR1
SCHEMBL8674849 0.84 CCR2 (0.48) TACR1
SCHEMBL8673624 0.84 TACR1 (0.46) TACR1
SCHEMBL8673191 0.84 TACR1 (0.48) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5696123-A ALPHA-PIPERAZINYL BENZYL COMPOUND AS TACHYKININ ANTAGONIST TREATING ASTHMA, BRONCHITIS, SKIN DISORDER, EYE DISEASE, HEADACHE, GASTROINTESTINAL DISORDER BOEHRINGER INGELHEIM KG (DE) 1997-12-09 US disclosed