SCHEMBL8919968

SCHEMBL8919968

COc1ccccc1C([CH]Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)N1CCN(C(c2ccccc2)c2ccccc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 10/20 0.47
CACNA2D1 P54289 2/20 0.43
CACNB1 Q02641 2/20 0.43
CACNA1A O00555 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
CYP3A4 P08684 1/20 0.41
CYP3A5 P20815 1/20 0.41
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
OPRL1 P41146 1/20 0.40
CACNA1B Q00975 1/20 0.39
CACNA1C Q13936 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8919912 0.91 TACR1 (0.46) TACR1
SCHEMBL8671580 0.89 TACR1 (0.49) TACR1
SCHEMBL8673617 0.89 TACR1 (0.49) TACR1
SCHEMBL8673323 0.88 TACR1 (0.47) TACR1
SCHEMBL8924107 0.87 TACR1 (0.46) TACR1MEN1KMT2A
SCHEMBL8673450 0.86 TACR1 (0.46) TACR1CACNA2D1CACNB1CACNA1AKMT2A
SCHEMBL8676401 0.85 KCNH2 (0.47) TACR1
SCHEMBL8673624 0.85 TACR1 (0.46) TACR1
SCHEMBL8674849 0.85 CCR2 (0.48) TACR1
SCHEMBL8673191 0.84 TACR1 (0.48) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5696123-A ALPHA-PIPERAZINYL BENZYL COMPOUND AS TACHYKININ ANTAGONIST TREATING ASTHMA, BRONCHITIS, SKIN DISORDER, EYE DISEASE, HEADACHE, GASTROINTESTINAL DISORDER BOEHRINGER INGELHEIM KG (DE) 1997-12-09 US disclosed