SCHEMBL8922608

SCHEMBL8922608

COc1cccc(C2C[C@@H](c3ccccc3)C[C@@H](N(C(N)=O)c3cccc(C)c3)C(=O)N2NC(=O)CC(C)(C)C)c1

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 15/20 0.40
GRIN2B Q13224 1/20 0.35
CHRNA7 P36544 2/20 0.34
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8922602 1.00 CCKBR (0.40) CCKBRGRIN2BCHRNA7PKM
SCHEMBL8922647 0.97 CCKBR (0.42) CCKBRGRIN2B
SCHEMBL8922643 0.97 CCKBR (0.42) CCKBRGRIN2B
SCHEMBL8921207 0.95 GRIN2B (0.37) CCKBRGRIN2BCHRNA7
SCHEMBL8921200 0.95 GRIN2B (0.37) CCKBRGRIN2BCHRNA7
SCHEMBL8919398 0.93 GRIN2B (0.38) CCKBRGRIN2B
SCHEMBL8919393 0.93 GRIN2B (0.38) CCKBRGRIN2B
SCHEMBL8922801 0.93 CCKBR (0.46) CCKBR
SCHEMBL8922812 0.93 CCKBR (0.46) CCKBR
SCHEMBL8922834 0.93 CCKBR (0.41) CCKBRGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5643904-A Substituted hexahdryoazepinones and tetrahydrobenzazepinones PFIZER INC. (US) 1997-07-01 US disclosed
US-5484917-A FOR TREATMENT AND PREVENTION OF GASTROINTESTINAL DISORDERS, PAIN AND ANXIETY PFIZER INC. (US) 1996-01-16 US disclosed