SCHEMBL8919398

SCHEMBL8919398

COc1cccc(N(C(N)=O)[C@@H]2C[C@@H](c3ccccc3)CC(c3ccccc3)N(NC(=O)CC(C)(C)C)C2=O)c1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 2/20 0.38
CCKBR P32239 11/20 0.37
OPRM1 P35372 1/20 0.37
MTNR1A P48039 1/20 0.35
MTNR1B P49286 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HSD17B1 P14061 1/20 0.34
HSD17B2 P37059 1/20 0.34
DGAT2 Q96PD7 1/20 0.34
ACHE P22303 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8919393 1.00 GRIN2B (0.38) GRIN2BCCKBROPRM1MTNR1AMTNR1B
SCHEMBL8921200 0.98 GRIN2B (0.37) GRIN2BCCKBROPRM1MTNR1AMTNR1B
SCHEMBL8921207 0.98 GRIN2B (0.37) GRIN2BCCKBROPRM1MTNR1AMTNR1B
SCHEMBL8922831 0.96 CCKBR (0.41) GRIN2BCCKBROPRM1MTNR1AMTNR1B
SCHEMBL8922834 0.96 CCKBR (0.41) GRIN2BCCKBROPRM1MTNR1AMTNR1B
SCHEMBL8920628 0.95 CCKBR (0.41) GRIN2BCCKBROPRM1SMN1; SMN2HSD17B1
SCHEMBL8920632 0.95 CCKBR (0.41) GRIN2BCCKBROPRM1SMN1; SMN2HSD17B1
SCHEMBL8922475 0.95 HSD17B1 (0.42) GRIN2BCCKBROPRM1MTNR1AMTNR1B
SCHEMBL8922479 0.95 HSD17B1 (0.42) GRIN2BCCKBROPRM1MTNR1AMTNR1B
SCHEMBL8922647 0.95 CCKBR (0.42) GRIN2BCCKBROPRM1MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5643904-A Substituted hexahdryoazepinones and tetrahydrobenzazepinones PFIZER INC. (US) 1997-07-01 US disclosed
US-5484917-A FOR TREATMENT AND PREVENTION OF GASTROINTESTINAL DISORDERS, PAIN AND ANXIETY PFIZER INC. (US) 1996-01-16 US disclosed