SCHEMBL8922669

SCHEMBL8922669

C[C@@H]1CN(C(=O)Nc2ccc3[nH]c(C(=O)N4CCN(c5ncccc5NC(C)(C)C)CC4)cc3c2)C[C@H](C)N1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.56
ADRA2A P08913 1/20 0.56
ADORA3 P0DMS8 1/20 0.56
CHRM1 P11229 1/20 0.56
MAOA P21397 1/20 0.56
TBXA2R P21731 1/20 0.56
OPRM1 P35372 1/20 0.56
MDH1 P40925 1/20 0.56
ABCG2 Q9UNQ0 1/20 0.56
TRPV1 Q8NER1 9/20 0.47
SYK P43405 7/20 0.43
NPSR1 Q6W5P4 1/20 0.43
HSD17B10 Q99714 1/20 0.43
TRPA1 O75762 1/20 0.41
TRPM8 Q7Z2W7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8923957 0.90 ADRA2A (0.70) KCNH2ADRA2AADORA3CHRM1MAOA
SCHEMBL9539638 0.82 ADRA2A (0.70) KCNH2ADRA2AADORA3CHRM1MAOA
SCHEMBL8923216 0.82 ADRA2A (0.70) KCNH2ADRA2AADORA3CHRM1MAOA
SCHEMBL8924496 0.81 ADRA2A (0.58) KCNH2ADRA2AADORA3CHRM1MAOA
SCHEMBL8794046 0.80 ADRA2A (0.73) KCNH2ADRA2AADORA3CHRM1MAOA
SCHEMBL8925498 0.79 ADRA2A (0.74) KCNH2ADRA2AADORA3CHRM1MAOA
SCHEMBL8922832 0.78 ADRA2A (0.68) KCNH2ADRA2AADORA3CHRM1MAOA
SCHEMBL8923782 0.78 ADRA2A (0.73) KCNH2ADRA2AADORA3CHRM1MAOA
SCHEMBL8921865 0.78 ADRA2A (0.72) KCNH2ADRA2AADORA3CHRM1MAOA
SCHEMBL8923448 0.77 ADRA2A (0.71) KCNH2ADRA2AADORA3CHRM1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5599930-A Substituted indoles as anti-AIDS pharmaceuticals THE UPJOHN COMPANY (US) 1997-02-04 US claimed
WO-1993001181-A1 SUBSTITUTED INDOLES AS ANTI-AIDS PHARMACEUTICALS THE UPJOHN COMPANY (US) 1993-01-21 WO claimed