SCHEMBL8923394

SCHEMBL8923394

COC(=O)c1c(Cl)cc(Cl)cc1NC(=S)CCCCc1cccs1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.41
KMT2A Q03164 5/20 0.41
GAA P10253 2/20 0.41
ALDH1A1 P00352 6/20 0.41
TSHR P16473 4/20 0.41
KDM4E B2RXH2 3/20 0.41
MAPK10 P53779 2/20 0.41
ALOX15 P16050 1/20 0.41
LMNA P02545 2/20 0.40
TDP1 Q9NUW8 2/20 0.39
L3MBTL1 Q9Y468 4/20 0.39
NPSR1 Q6W5P4 3/20 0.39
MAPK1 P28482 2/20 0.39
GLA P06280 1/20 0.39
BLM P54132 1/20 0.38
CTDSP1 Q9GZU7 1/20 0.38
MAPK8 P45983 1/20 0.38
MAPK9 P45984 1/20 0.38
POLB P06746 3/20 0.38
DNMT1 P26358 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8921856 0.82 POLB (0.41) MEN1KMT2AGAAALDH1A1TSHR
SCHEMBL8922395 0.81 CYP4A11 (0.47) MEN1KMT2AGAAALDH1A1ALOX15
SCHEMBL8923389 0.80 ALDH1A1 (0.43) MEN1KMT2AGAAALDH1A1TSHR
SCHEMBL8921268 0.80 CYP4F2 (0.52) MEN1KMT2AGAAALDH1A1MAPT
SCHEMBL8921195 0.78 MAPT (0.48) MEN1KMT2AGAAALDH1A1L3MBTL1
SCHEMBL8921377 0.77 ALDH1A1 (0.46) MEN1KMT2AALDH1A1KDM4ELMNA
SCHEMBL6331207 0.70 SMN1; SMN2 (0.62) ALDH1A1TSHRL3MBTL1POLBSMN1; SMN2
SCHEMBL8921612 0.69 SMN1; SMN2 (0.37) KMT2AALDH1A1TSHRKDM4ELMNA
SCHEMBL8922762 0.69 MALT1 (0.48) TSHRLMNAPOLBHTTMAPT
SCHEMBL11792109 0.69 SMN1; SMN2 (0.61) ALDH1A1TSHRL3MBTL1POLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633379-A N-METHYLASPARTIC ACID ANTAGONIST CIBA-GEIGY CORPORATION (US) 1997-05-27 US disclosed
EP-0685466-A1 3-Heteroaliphatyle-and 3-hetero-(aryle)-aliphatyle-2(1H)-quinolone derivatives CIBA-GEIGY AG (CH) 1995-12-06 EP disclosed