SCHEMBL8924501

SCHEMBL8924501

O=C(c1ccccc1)C1CCCN=N1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.44
CPB1 P15086 1/20 0.38
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
HTT P42858 2/20 0.37
MAPT P10636 1/20 0.37
ALOX15 P16050 1/20 0.37
HBB P68871 1/20 0.37
SLC18A3 Q16572 2/20 0.36
EPHX1 P07099 1/20 0.36
HTR2A P28223 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ATM Q13315 1/20 0.35
DAO P14920 1/20 0.34
TSHR P16473 1/20 0.34
NAPRT Q6XQN6 1/20 0.34
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2646530 0.82 MCL1 (0.46) MCL1CPB1NPC1RAB9AHTT
SCHEMBL1624945 0.77 MCL1 (0.49) MCL1NPC1RAB9AHTTMAPT
SCHEMBL9041510 0.69 SRD5A2 (0.47) MCL1CPB1SLC18A3HTR2AMEN1
SCHEMBL27848887 0.69 MCL1 (0.51) MCL1CPB1HTTMAPTALOX15
SCHEMBL7295695 0.69 MCL1 (0.44) MCL1CPB1MAPTSLC18A3HTR2A
SCHEMBL30484842 0.68 MEN1 (0.56) MAPTMEN1KMT2A
SCHEMBL965420 0.67 SRD5A2 (0.63) MCL1CPB1SLC18A3HTR2AMEN1
SCHEMBL9920449 0.67 MCL1 (0.58) MCL1NPC1RAB9AHTTMAPT
SCHEMBL3113279 0.67 SRD5A2 (0.58) MCL1CPB1SLC18A3HTR2AMEN1
SCHEMBL654047 0.67 HTR2A (0.49) MCL1CPB1SLC18A3HTR2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5684151-A PROGESTIN AGONISTS ORTHO PHARMACEUTICAL CORPORATION (US) 1997-11-04 US disclosed
EP-0650480-A1 1-ARYLSULPHONYL, ARYLCARBONYL AND 1-ARYLPHOSPHONYL-3-PHENYL-1,4,5,6-TETRAHYDROPYRIDAZINES ORTHO PHARMACEUTICAL CORPORATION (US) 1995-05-03 EP disclosed
WO-1994001412-A1 1-ARYLSULPHONYL, ARYLCARBONYL AND 1-ARYLPHOSPHONYL-3-PHENYL-1,4,5,6-TETRAHYDROPYRIDAZINES ORTHO PHARMACEUTICAL CORPORATION (US) 1994-01-20 WO disclosed