SCHEMBL8925823

SCHEMBL8925823

CCCNc1cccnc1N1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.49
POLB P06746 1/20 0.49
KIT P10721 2/20 0.47
TRPA1 O75762 3/20 0.47
TRPV1 Q8NER1 2/20 0.47
CKS1B P61024 2/20 0.46
SKP1 P63208 2/20 0.46
SKP2 Q13309 2/20 0.46
GPR119 Q8TDV5 3/20 0.46
DTYMK P23919 1/20 0.45
GBA1 P04062 1/20 0.45
HTR3E A5X5Y0 1/20 0.45
HTR3B O95264 1/20 0.45
HTR3A P46098 1/20 0.45
HTR3D Q70Z44 1/20 0.45
HTR3C Q8WXA8 1/20 0.45
GAA P10253 1/20 0.43
GRIA1 P42261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28766136 0.93 ACHE (0.47) ACHEPOLBKITTRPA1TRPV1
SCHEMBL3330474 0.91 POLB (0.51) ACHEPOLBKITTRPA1TRPV1
SCHEMBL8794748 0.87 POLB (0.49) ACHEPOLBKITTRPA1TRPV1
SCHEMBL31652137 0.85 POLB (0.54) ACHEPOLBKITTRPA1TRPV1
SCHEMBL8923840 0.85 ACHE (0.48) ACHEPOLBKITTRPA1TRPV1
SCHEMBL22587512 0.83 POLB (0.52) ACHEPOLBKITTRPA1TRPV1
SCHEMBL8921494 0.83 POLB (0.47) ACHEPOLBKITTRPA1TRPV1
SCHEMBL29741439 0.82 POLB (0.54) ACHEPOLBKITTRPA1TRPV1
SCHEMBL8793643 0.82 POLB (0.54) ACHEPOLBKITTRPA1TRPV1
SCHEMBL31652019 0.82 POLB (0.55) ACHEPOLBKITTRPA1TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5599930-A Substituted indoles as anti-AIDS pharmaceuticals THE UPJOHN COMPANY (US) 1997-02-04 US disclosed
US-5563142-A INHIBITORS OF VIRAL REVERSE TRANSCRIPTASE THE UPJOHN COMPANY (US) 1996-10-08 US disclosed
EP-0507861-B1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS UPJOHN CO (US) 1996-09-11 EP disclosed
US-5489593-A Anti-aids piperazines THE UPJOHN COMPANY (US) 1996-02-06 US disclosed
WO-1993001181-A1 SUBSTITUTED INDOLES AS ANTI-AIDS PHARMACEUTICALS THE UPJOHN COMPANY (US) 1993-01-21 WO disclosed
EP-0507861-A1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS. UPJOHN CO (US) 1992-10-14 EP disclosed