SCHEMBL8925912

SCHEMBL8925912

Cc1nc(-c2cc(C)c(OCCCc3cnc4ccccc4c3)c(C)c2)no1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
HDAC6 Q9UBN7 1/20 0.41
L3MBTL1 Q9Y468 6/20 0.39
PDE10A Q9Y233 4/20 0.38
TDP1 Q9NUW8 3/20 0.37
ATM Q13315 1/20 0.37
CYP1A2 P05177 1/20 0.35
MAPT P10636 3/20 0.35
TSHR P16473 3/20 0.35
LMNA P02545 3/20 0.35
DRD2 P14416 1/20 0.35
MAPK1 P28482 4/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
CFTR P13569 1/20 0.34
HPGD P15428 1/20 0.34
CASP3 P42574 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8925641 0.87 NR1I2 (0.64) NR1I2CYP3A4CYP2D6HDAC6
SCHEMBL8921466 0.81 NR1I2 (0.45) NR1I2CYP3A4CYP2D6L3MBTL1TDP1
SCHEMBL8924593 0.80 CYP3A4 (0.44) NR1I2CYP3A4CYP2D6HDAC6L3MBTL1
SCHEMBL9200266 0.76 NR1I2 (0.73) NR1I2CYP3A4CYP2D6L3MBTL1TDP1
SCHEMBL8824399 0.76 NR1I2 (0.52) NR1I2CYP3A4CYP2D6L3MBTL1TDP1
SCHEMBL9087864 0.74 NR1I2 (0.47) NR1I2CYP3A4CYP2D6L3MBTL1TDP1
SCHEMBL8824422 0.74 NR1I2 (0.53) NR1I2CYP3A4CYP2D6L3MBTL1TDP1
SCHEMBL8670645 0.74 CYP3A4 (0.48) NR1I2CYP3A4CYP2D6L3MBTL1TDP1
SCHEMBL8553518 0.74 NR1I2 (0.49) NR1I2CYP3A4CYP2D6L3MBTL1TDP1
SCHEMBL8824435 0.73 NR1I2 (0.49) NR1I2CYP3A4CYP2D6HDAC6L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5618821-A VIRICIDES, PICORNAVIRUS SANOFI, S.A. (FR) 1997-04-08 US disclosed
WO-1995031438-A1 THERAPEUTIC PHENOXYALKYLHETEROCYCLES SANOFI WINTHROP, INC. (US) 1995-11-23 WO disclosed