SCHEMBL8926094

SCHEMBL8926094

CCOC(=O)c1nc(C(=O)CBr)ccc1O

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.46
CA12 O43570 5/20 0.44
CA1 P00915 5/20 0.44
CA2 P00918 5/20 0.44
CA7 P43166 5/20 0.44
CA9 Q16790 5/20 0.44
CA14 Q9ULX7 5/20 0.44
NPC1 O15118 6/20 0.42
RAB9A P51151 4/20 0.42
ALDH1A1 P00352 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
TARBP2 Q15633 2/20 0.41
KDM4E B2RXH2 2/20 0.40
LMNA P02545 1/20 0.40
HSD17B2 P37059 1/20 0.40
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40
NR1H2 P55055 1/20 0.39
NR1H3 Q13133 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL5434830 0.98 CYP1A2 (0.45) CYP1A2CA12CA1CA2CA7
SCHEMBL1301427 0.78 CYP1A2 (0.77) CYP1A2CA12CA1CA2CA7
SCHEMBL31236724 0.78 CA12 (0.49) CYP1A2CA12CA1CA2CA7
SCHEMBL25248606 0.78 CA12 (0.49) CYP1A2CA12CA1CA2CA7
SCHEMBL8922334 0.74 CYP1A2 (0.51) CYP1A2CA12CA1CA2CA7
SCHEMBL18132220 0.73 CYP1A2 (0.59) CYP1A2NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL6202564 0.72 CYP1A2 (0.53) CYP1A2NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL27972725 0.72 MAPT (0.50) CYP1A2CA12CA1CA2CA7
SCHEMBL6201965 0.71 POLB (0.47) CYP1A2NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL16600772 0.70 GRIN2B (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5639770-A SUPEROXIDE INHIBITOR OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-06-17 US disclosed
EP-0600092-A1 THIAZOLE DERIVATIVE OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-06-08 EP disclosed