SCHEMBL8926496

SCHEMBL8926496

CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CC4CCOC4(CNC(=O)OC(C)(C)C)C3)c(F)c21

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.49
HSD17B10 Q99714 6/20 0.49
ALDH1A1 P00352 5/20 0.49
HPGD P15428 5/20 0.49
PMP22 Q01453 1/20 0.49
KCNH2 Q12809 3/20 0.38
DRD3 P35462 1/20 0.37
BRD4 O60885 1/20 0.36
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.36
CYP2J2 P51589 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
KMT2A Q03164 1/20 0.36
TOP1 P11387 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9210491 0.92 KDM4E (0.40) KDM4EHSD17B10ALDH1A1HPGDPMP22
SCHEMBL7836509 0.90 KCNH2 (0.46) KDM4EHSD17B10ALDH1A1HPGDKCNH2
SCHEMBL7846922 0.90 KCNH2 (0.46) KDM4EHSD17B10ALDH1A1HPGDKCNH2
SCHEMBL7846924 0.90 KCNH2 (0.46) KDM4EHSD17B10ALDH1A1HPGDKCNH2
SCHEMBL7492274 0.90 KDM4E (0.38) KDM4EHSD17B10ALDH1A1HPGDPMP22
SCHEMBL7494366 0.90 KCNH2 (0.46) KDM4EHSD17B10ALDH1A1HPGDKCNH2
SCHEMBL7836504 0.90 KCNH2 (0.46) KDM4EHSD17B10ALDH1A1HPGDKCNH2
SCHEMBL8925166 0.88 CYP3A4 (0.39) KDM4EHSD17B10ALDH1A1HPGDPMP22
SCHEMBL8925167 0.88 CYP3A4 (0.39) KDM4EHSD17B10ALDH1A1HPGDPMP22
SCHEMBL8922822 0.85 ALDH1A1 (0.51) KDM4EHSD17B10ALDH1A1HPGDKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5621105-A REACTING HALO-SUBSTITUTED QUINOLONECARBOXYLIC ACID OR NAPHTHYRIDONECARBOXYLIC ACID WITH 1-AMINOMETHYL-2-OXA-7-AZABICYCLO/3.3.0/OCTANE BAYER AKTIENGESELLSCHAFT (DE) 1997-04-15 US disclosed
US-5574161-A GRAMPOSITIVE BACTERICIDE BAYER AKTIENGESELLSCHAFT (DE) 1996-11-12 US disclosed
EP-0589318-B1 Antibacterial 7-(aminomethyl-oxa-7-azabicyclo(3.3.0)oct-7-yl)quinolone- and -naphthyridonecarboxylic acid derivatives BAYER AG (DE) 1995-11-15 EP disclosed
US-5395944-A Bactericides BAYER AKTIENGESELLSCHAFT (DE) 1995-03-07 US disclosed
EP-0589318-A2 Antibacterial 7-(aminomethyl-oxa-7-azabicyclo(3.3.0)oct-7-yl)quinolone- and -naphthyridonecarboxylic acid derivatives BAYER AG (DE) 1994-03-30 EP disclosed