SCHEMBL9210491

SCHEMBL9210491

CCn1cc(OC(=O)O)c(=O)c2cc(F)c(N3CC4CCOC4(CNC(=O)OC(C)(C)C)C3)c(F)c21

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.40
ALDH1A1 P00352 4/20 0.40
HPGD P15428 4/20 0.40
HSD17B10 Q99714 3/20 0.40
PMP22 Q01453 1/20 0.39
KCNH2 Q12809 1/20 0.31
MEN1 O00255 1/20 0.30
GAA P10253 1/20 0.30
KMT2A Q03164 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8926496 0.92 KDM4E (0.49) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL7494369 0.90 KCNH2 (0.37) KDM4EALDH1A1HPGDHSD17B10KCNH2
SCHEMBL7496654 0.90 KCNH2 (0.37) KDM4EALDH1A1HPGDHSD17B10KCNH2
SCHEMBL7501610 0.90 KCNH2 (0.37) KDM4EALDH1A1HPGDHSD17B10KCNH2
SCHEMBL7492282 0.90 KDM4E (0.31) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9209492 0.89 CYP3A4 (0.31) KCNH2
SCHEMBL9214867 0.86 ALDH1A1 (0.42) KDM4EALDH1A1HPGDHSD17B10KCNH2
Hydrochloric Acid SCHEMBL9210346 0.85 KDM4E (0.45) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL7493085 0.85 KCNH2 (0.45) KDM4EALDH1A1HPGDHSD17B10KCNH2
SCHEMBL9274990 0.85 KDM4E (0.44) KDM4EALDH1A1HPGDHSD17B10KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0520674-B1 Antipsychotic benzodioxan derivatives AMERICAN HOME PROD (US) 1995-08-16 EP claimed