SCHEMBL8927740

SCHEMBL8927740

[CH2]c1cn(O)c2ccccc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR3 P46089 1/20 0.36
CYP2C19 P33261 2/20 0.34
CYP1A2 P05177 1/20 0.34
POLB P06746 1/20 0.34
KDM4E B2RXH2 6/20 0.33
ALDH1A1 P00352 3/20 0.33
BACE1 P56817 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
HTT P42858 2/20 0.33
GLA P06280 2/20 0.33
ERCC1 P07992 1/20 0.33
FEN1 P39748 1/20 0.33
ERCC4 Q92889 1/20 0.33
CCNT1 O60563 1/20 0.33
CDK9 P50750 1/20 0.33
ATM Q13315 1/20 0.33
P2RX4 Q99571 1/20 0.33
MAPK1 P28482 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9654009 0.74 IDO1 (0.42) GPR3CYP2C19CYP1A2POLBKDM4E
SCHEMBL28562457 0.73 GPR3 (0.36) GPR3CYP2C19CYP1A2POLBKDM4E
SCHEMBL8927744 0.73 MEN1 (0.46) GPR3CYP2C19CYP1A2POLBKDM4E
SCHEMBL315328 0.73 GPR84 (0.55) GPR3POLBKDM4EALDH1A1HTT
SCHEMBL8186050 0.72 ASH1L (0.47) CYP2C19CYP1A2POLBKDM4EALDH1A1
SCHEMBL20674511 0.71 GPR84 (0.44) GPR3CYP2C19CYP1A2POLBKDM4E
SCHEMBL887129 0.71 HTT (0.54) POLBKDM4EALDH1A1HTTGLA
SCHEMBL8530588 0.71 KDM4E (0.41) POLBKDM4EALDH1A1HTTMEN1
SCHEMBL9550626 0.70 CYP1A2 (0.37) CYP1A2POLBKDM4EALDH1A1L3MBTL1
SCHEMBL8527729 0.70 POLB (0.33) GPR3POLBKDM4EALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5614498-A OLIGOPEPTIDES, BRONCHDILATORS BANYU PHARMACEUTICAL CO., LTD. (JP) 1997-03-25 US disclosed
US-5496928-A Endothelin antagonistic substance BANYU PHARMACEUTICAL CO., LTD. (JP) 1996-03-05 US disclosed
EP-0555537-A2 Endothelin antagonistic substance BANYU PHARMACEUTICAL CO., LTD. (JP) 1993-08-18 EP disclosed