SCHEMBL8928369

SCHEMBL8928369

CC(C)(C)OC(=O)CN(CCN(CC(=O)OC(C)(C)C)CC(=O)OC(C)(C)C)CCN(CC(=O)OC(C)(C)C)C(COCc1ccc(NC(=O)CNC(=O)OC(C)(C)C)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 2/20 0.36
EGFR P00533 2/20 0.35
AURKB Q96GD4 2/20 0.35
MAPT P10636 3/20 0.35
TDP1 Q9NUW8 3/20 0.35
PPARG P37231 1/20 0.35
LTA4H P09960 1/20 0.35
CTSS P25774 1/20 0.34
TLR7 Q9NYK1 1/20 0.34
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
PABPC1 P11940 1/20 0.33
XBP1 P17861 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
GPR55 Q9Y2T6 1/20 0.33
PTPRB P23467 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8928353 0.82 PPARA (0.36) PPARAPPARGCTSSCA1CA2
SCHEMBL8928375 0.79 NR1D1 (0.47) PPARAMAPTPPARG
SCHEMBL8059351 0.78 PPARA (0.46) PPARAPPARGCTSSNPSR1L3MBTL1
SCHEMBL8387845 0.77
SCHEMBL6432521 0.74 PPARA (0.43) PPARAPPARGLTA4HCTSSCA1
SCHEMBL6429868 0.72 PPARA (0.43) PPARAPPARGLTA4HCTSSCA1
SCHEMBL8693590 0.71 CA1 (0.54) EGFRAURKBMAPTTDP1TLR7
SCHEMBL23572300 0.69 EPOR (0.41) PPARACTSSCA1CA2SMN1; SMN2
SCHEMBL7666444 0.69 ATM (0.40) MAPTTDP1CTSSCA1
SCHEMBL7511620 0.69 CTSS (0.40) CTSSCA1CA2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5649537-A CONJUGATION OF A BILE ACID WITH A CHELATING AGENT AND BI- OR TRIVALENT METALS; IMAGING OF THE HEPTATOBILIARY SYSTEM; NUCLEAR MAGNETIC RESONANCE DIBRA S.P.A. (IT) 1997-07-22 US disclosed