SCHEMBL8929209

SCHEMBL8929209

c1nc(Nc2ccc3c(c2)CCC3)c2cc[nH]c2n1

nearest known ligand 0.63

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.63
TTBK1 Q5TCY1 15/20 0.58
TTBK2 Q6IQ55 15/20 0.58
AURKA O14965 1/20 0.56
AURKB Q96GD4 1/20 0.56
INCENP Q9NQS7 1/20 0.56
LCK P06239 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8928980 0.99 EGFR (0.62) EGFRTTBK1TTBK2AURKAAURKB
SCHEMBL8929392 0.81 EGFR (0.58) EGFRTTBK1TTBK2AURKAAURKB
Hydrochloric Acid SCHEMBL8929775 0.80 EGFR (0.57) EGFRTTBK1TTBK2AURKAAURKB
SCHEMBL23408992 0.76 TTBK1 (0.62) EGFRTTBK1TTBK2AURKAAURKB
SCHEMBL8929171 0.76 BCL6 (0.60) EGFRTTBK1TTBK2AURKAAURKB
Hydrochloric Acid SCHEMBL8929519 0.75 BCL6 (0.58) EGFRTTBK1TTBK2AURKAAURKB
SCHEMBL7021509 0.75 EGFR (0.70) EGFRTTBK1TTBK2AURKAAURKB
SCHEMBL7832906 0.75 EGFR (0.59) EGFRLCK
Hydrochloric Acid SCHEMBL7020471 0.74 EGFR (0.69) EGFRTTBK1TTBK2AURKAAURKB
SCHEMBL16363320 0.74 TTBK1 (0.84) TTBK1TTBK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0795556-A1 4-Substituted pyrrolopyrimidine compounds as tyrosin kinase inhibitors PHARMACIA & UPJOHN S.p.A. (IT) 1997-09-17 EP claimed
EP-0795556-A1 4-Substituted pyrrolopyrimidine compounds as tyrosin kinase inhibitors PHARMACIA & UPJOHN S.p.A. (IT) 1997-09-17 EP disclosed