SCHEMBL8929293

SCHEMBL8929293

c1ccc2c(c1)CCC(Oc1ncnc3[nH]ccc13)C2

nearest known ligand 0.62

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 6/20 0.62
TRPA1 O75762 5/20 0.49
JAK2 O60674 4/20 0.43
JAK1 P23458 3/20 0.43
HPGDS O60760 1/20 0.39
HTR2C P28335 1/20 0.39
SLC6A4 P31645 1/20 0.39
HTR2B P41595 1/20 0.39
TTBK1 Q5TCY1 1/20 0.38
TTBK2 Q6IQ55 1/20 0.38
KIT P10721 1/20 0.38
AKT2 P31751 1/20 0.38
GSK3B P49841 1/20 0.38
NUDT1 P36639 1/20 0.38
IDO1 P14902 1/20 0.37
TYK2 P29597 2/20 0.37
BMX P51813 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3532381 0.77 JAK3 (1.00) JAK3TRPA1JAK2JAK1HPGDS
SCHEMBL20183342 0.76 JAK3 (0.76) JAK3TRPA1JAK2JAK1HPGDS
SCHEMBL8929492 0.76 JAK3 (0.56) JAK3TRPA1JAK2JAK1HPGDS
SCHEMBL1980392 0.75 JAK3 (0.74) JAK3TRPA1JAK2JAK1HPGDS
SCHEMBL8929835 0.73 HPGDS (0.63) JAK3JAK1HPGDSTTBK1TTBK2
SCHEMBL8929626 0.72 CYP19A1 (0.46) JAK3JAK2JAK1HPGDSTTBK1
Hydrochloric Acid SCHEMBL8929253 0.72 HPGDS (0.61) JAK3JAK1HPGDSTTBK1TTBK2
SCHEMBL8929274 0.72 CDC7 (0.46) JAK3TRPA1JAK2JAK1HPGDS
SCHEMBL17545945 0.72 JAK3 (0.73) JAK3TRPA1JAK2JAK1HPGDS
SCHEMBL3530525 0.72 JAK1 (0.67) JAK3JAK2JAK1TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0795556-A1 4-Substituted pyrrolopyrimidine compounds as tyrosin kinase inhibitors PHARMACIA & UPJOHN S.p.A. (IT) 1997-09-17 EP claimed
EP-0795556-A1 4-Substituted pyrrolopyrimidine compounds as tyrosin kinase inhibitors PHARMACIA & UPJOHN S.p.A. (IT) 1997-09-17 EP disclosed