SCHEMBL892990

SCHEMBL892990

Cc1nc(-c2ccccc2)sc1C(=O)Cl

nearest known ligand 0.76

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 7/20 0.76
ALDH1A1 P00352 6/20 0.70
MAPT P10636 6/20 0.70
GAA P10253 3/20 0.70
HPGD P15428 2/20 0.69
NPSR1 Q6W5P4 1/20 0.69
NPC1 O15118 4/20 0.62
RAB9A P51151 6/20 0.61
KMT2A Q03164 3/20 0.61
LMNA P02545 2/20 0.61
ATM Q13315 1/20 0.61
KDM4E B2RXH2 2/20 0.60
POLB P06746 1/20 0.60
L3MBTL1 Q9Y468 3/20 0.59
MEN1 O00255 2/20 0.59
CNR1 P21554 2/20 0.57
NPY1R P25929 1/20 0.56
NPY2R P49146 1/20 0.56
TDP1 Q9NUW8 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10223891 0.87 SMN1; SMN2 (0.76) SMN1; SMN2ALDH1A1MAPTGAAHPGD
SCHEMBL1327631 0.86 SMN1; SMN2 (1.00) SMN1; SMN2ALDH1A1MAPTGAAHPGD
SCHEMBL12475206 0.85 SMN1; SMN2 (0.77) SMN1; SMN2ALDH1A1MAPTGAAHPGD
SCHEMBL851866 0.85 SMN1; SMN2 (0.78) SMN1; SMN2ALDH1A1MAPTGAAHPGD
SCHEMBL28795980 0.84 RAB9A (0.57) SMN1; SMN2ALDH1A1MAPTGAAHPGD
SCHEMBL289112 0.83 SMN1; SMN2 (0.93) SMN1; SMN2ALDH1A1MAPTGAAHPGD
SCHEMBL4243016 0.83 SMN1; SMN2 (0.76) SMN1; SMN2ALDH1A1MAPTGAAHPGD
SCHEMBL3065347 0.83 CYP1A2 (0.75) SMN1; SMN2ALDH1A1MAPTGAAHPGD
SCHEMBL3068544 0.83 SMN1; SMN2 (0.60) SMN1; SMN2ALDH1A1MAPTGAANPC1
Hydrochloric Acid SCHEMBL11388173 0.82 CYP1A2 (0.73) SMN1; SMN2ALDH1A1MAPTGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 55 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119638737-A Macrocyclic compounds and their use in medicine 广东东阳光药业股份有限公司 2025-03-18 CN disclosed
CN-107089993-B Hypolipidemic activity bamboo-cypress lactone compound, preparation method and application thereof 中国科学院上海药物研究所 2024-07-09 CN disclosed
EP-3190109-B1 INDOLE AMIDE DERIVATIVES AND RELATED COMPOUNDS FOR USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES UNIV LEUVEN KATH (BE) 2020-02-19 EP disclosed
US-20190054068-A1 Indole Amide Derivatives and Related Compounds for Use in the Treatment of Neurodegenerative Diseases REMYND (BE) 2019-02-21 US disclosed
US-10117850-B2 Indole amide derivatives and related compounds for use in the treatment of neurodegenerative diseases KATHOLIEKE UNIVERSITEIT LEUVEN, K.U.LEUVEN R&D (BE) 2018-11-06 US disclosed
EP-3190109-A1 INDOLE AMIDE DERIVATIVES AND RELATED COMPOUNDS FOR USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES Katholieke Universiteit Leuven (BE) 2017-07-12 EP disclosed
EP-2440550-B1 INDOLE AMIDE DERIVATIVES AND RELATED COMPOUNDS FOR USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES UNIV LEUVEN KATH (BE) 2017-03-15 EP disclosed
US-20160324828-A1 INDOLE AMIDE DERIVATIVES AND RELATED COMPOUNDS FOR USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES KATHOLIEKE UNIVERSITEIT LEUVEN, K.U.LEUVEN R&D (BE) 2016-11-10 US disclosed
US-9434722-B2 Indole amide derivatives and related compounds for use in the treatment of neurodegenerative diseases KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2016-09-06 US disclosed
CN-102532123-B Thiazole-5-methanamide compound and method for making thereof and pharmaceutical composition and purposes INSTITUTE OF MATARIA MEDICA, CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2016-03-09 CN disclosed
CN-100363348-C PgD2 receptor antagonists for the treatment of inflammatory diseases MILLENNIUM PHARM INC (US) 2008-01-23 CN disclosed
CN-101018770-A PGD2 receptor antagonists for the treatment of inflammatory diseases MILLENNIUM PHARM INC (US) 2007-08-15 CN disclosed
US-7211672-B2 PGD2 receptor antagonists for the treatment of inflammatory diseases MILLENNIUM PHARMACEUTICALS, INC. (US) 2007-05-01 US disclosed
US-20070049618-A1 Isoindole-imide compounds and compositions comprising and methods of using the same CELGENE CORPORATION 2007-03-01 US disclosed
US-20060106061-A1 PGD2 receptor antagonists for the treatment of inflammatory diseases MILLENNIUM PHARMACEUTICALS, INC. 2006-05-18 US disclosed
CN-1720047-A PgD2 receptor antagonists for the treatment of inflammatory diseases MILLENNIUM PHARM INC (US) 2006-01-11 CN disclosed
US-20050256158-A1 PGD2 receptor antagonists for the treatment of inflammatory diseases MILLENNIUM PHARMACEUTICALS, INC. 2005-11-17 US disclosed
US-20050222160-A1 Thiazole derivatives as phosphodiesterase iv inhibitors MERCK PATENT GMBH (DE) 2005-10-06 US disclosed
CN-1662529-A Thiazole derivatives as phosphodiesterase IV inhibitors MERCK PATENT GMBH (DE) 2005-08-31 CN disclosed
US-20040082609-A1 PGD2 receptor antagonists for the treatment of inflammatory diseases MILLENNIUM PHARMACEUTICALS, INC. 2004-04-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160324828-A1 INDOLE AMIDE DERIVATIVES AND RELATED COMPOUNDS FOR USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES SNCA, MAPT, NLN SMN1; SMN2 81/4885ALDH1A1 2404/4885MAPT 2/4885
US-20050256158-A1 PGD2 receptor antagonists for the treatment of inflammatory diseases PTGDR2, LTB4R2, CYSLTR2 SMN1; SMN2 4770/4885ALDH1A1 1599/4885MAPT 4208/4885
US-20060106061-A1 PGD2 receptor antagonists for the treatment of inflammatory diseases PTGDR2, LTB4R2, CYSLTR2 SMN1; SMN2 4803/4885ALDH1A1 2039/4885MAPT 4401/4885
US-20190054068-A1 Indole Amide Derivatives and Related Compounds for Use in the Treatment of Neurodegenerative Diseases SNCA, MAPT, NLN SMN1; SMN2 80/4885ALDH1A1 2395/4885MAPT 2/4885
US-10117850-B2 Indole amide derivatives and related compounds for use in the treatment of neurodegenerative diseases SNCA, MAPT, NLN SMN1; SMN2 81/4885ALDH1A1 2404/4885MAPT 2/4885
US-20050222160-A1 Thiazole derivatives as phosphodiesterase iv inhibitors PDE3B, PDE4B, PDE4A SMN1; SMN2 3019/4885ALDH1A1 1542/4885MAPT 4552/4885
US-20070049618-A1 Isoindole-imide compounds and compositions comprising and methods of using the same SI, CYP3A5, CYP2D6 SMN1; SMN2 1271/4885ALDH1A1 1081/4885MAPT 553/4885
US-20040082609-A1 PGD2 receptor antagonists for the treatment of inflammatory diseases PTGDR2, PTGDR, LTB4R2 SMN1; SMN2 4763/4885ALDH1A1 1663/4885MAPT 4629/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.