SCHEMBL8930446

SCHEMBL8930446

CCN(CC)C(=O)c1cccc(C(c2cccc(O)c2)N2CC(C)NCC2C)c1

nearest known ligand 0.68

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.58
OPRD1 P41143 2/20 0.58
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2C9 P11712 1/20 0.58
HPGD P15428 1/20 0.58
OPRK1 P41145 1/20 0.58
SIGMAR1 Q99720 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8930430 1.00 OPRM1 (0.58) OPRM1OPRD1CYP1A2CYP3A4CYP2C9
SCHEMBL8930437 1.00 OPRM1 (0.58) OPRM1OPRD1CYP1A2CYP3A4CYP2C9
SCHEMBL236139 0.93 OPRD1 (0.67) OPRM1OPRD1CYP1A2CYP3A4CYP2C9
SCHEMBL236138 0.93 OPRD1 (0.67) OPRM1OPRD1CYP1A2CYP3A4CYP2C9
SCHEMBL4576571 0.93 OPRD1 (0.67) OPRM1OPRD1CYP1A2CYP3A4CYP2C9
SCHEMBL233715 0.93 OPRD1 (0.67) OPRM1OPRD1CYP1A2CYP3A4CYP2C9
SCHEMBL4575467 0.93 OPRD1 (0.67) OPRM1OPRD1CYP1A2CYP3A4CYP2C9
SCHEMBL4575507 0.93 OPRD1 (0.67) OPRM1OPRD1CYP1A2CYP3A4CYP2C9
SCHEMBL18661816 0.93 OPRD1 (0.67) OPRM1OPRD1CYP1A2CYP3A4CYP2C9
SCHEMBL233716 0.93 OPRD1 (0.67) OPRM1OPRD1CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5681830-A DIARYLMETHYL PIPERAZINE COMPOUNDS HAVING UTILITY IN MEDICAL THERAPY AS RECEPTOR-BINDING SPECIES DELTA PHARMACEUTICALS, INC. (US) 1997-10-28 US disclosed