Terephthalamide

Terephthalamide

SCHEMBL8931235

NC(=O)c1ccc(C(N)=O)cc1.NCN

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.60
TSHR P16473 2/20 0.60
POLB P06746 1/20 0.60
CYP3A4 P08684 1/20 0.60
MAPT P10636 1/20 0.60
CYP2C19 P33261 1/20 0.60
RECQL P46063 1/20 0.60
BLM P54132 1/20 0.60
PMP22 Q01453 1/20 0.60
HSD17B10 Q99714 1/20 0.60
TDP1 Q9NUW8 1/20 0.60
L3MBTL1 Q9Y468 1/20 0.60
PARP10 Q53GL7 12/20 0.59
PARP4 Q9UKK3 2/20 0.59
PARP15 Q460N3 2/20 0.59
ALDH1A1 P00352 1/20 0.59
KMT2A Q03164 1/20 0.59
PARP14 Q460N5 1/20 0.59
PARP16 Q8N5Y8 1/20 0.59
PARP11 Q9NR21 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Terephthalamide SCHEMBL23774 0.90 PARP1 (0.71) PARP1TSHRPOLBCYP3A4MAPT
Terephthalamide SCHEMBL28360111 0.87 PARP1 (0.67) PARP1TSHRPOLBCYP3A4MAPT
Terephthalamide SCHEMBL29102653 0.87 PARP1 (0.67) PARP1TSHRPOLBCYP3A4MAPT
Terephthalamide SCHEMBL27281597 0.87 PARP1 (0.67) PARP1TSHRPOLBCYP3A4MAPT
Terephthalamide SCHEMBL11512422 0.87 PARP1 (0.67) PARP1TSHRPOLBCYP3A4MAPT
Terephthalamide SCHEMBL689841 0.87 PARP1 (0.67) PARP1TSHRPOLBCYP3A4MAPT
Terephthalamide SCHEMBL1906838 0.87 PARP1 (0.67) PARP1TSHRPOLBCYP3A4MAPT
Terephthalamide SCHEMBL1087289 0.87 PARP1 (0.67) PARP1TSHRPOLBCYP3A4MAPT
Terephthalamide SCHEMBL15328883 0.87 PARP1 (0.67) PARP1TSHRPOLBCYP3A4MAPT
Terephthalamide SCHEMBL7508927 0.87 PARP1 (0.67) PARP1TSHRPOLBCYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0753027-A1 THERMOPLASTIC ELASTOMERS HAVING IMPROVED SURFACE PROPERTIES ADVANCED ELASTOMER SYSTEMS (US) 1997-01-15 EP disclosed
WO-1995026380-A1 THERMOPLASTIC ELASTOMERS HAVING IMPROVED SURFACE PROPERTIES ADVANCED ELASTOMER SYSTEMS, L.P. (US) 1995-10-05 WO disclosed
EP-0436080-A2 Core-shell polymer and its use Takeda Chemical Industries, Ltd. (JP) 1991-07-10 EP disclosed
EP-0423628-A2 Core-shell polymer, resin composition and molded article thereof Takeda Chemical Industries, Ltd. (JP) 1991-04-24 EP disclosed
EP-0258040-A1 Thermoplastic resin composition comprising a polyamide SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1988-03-02 EP disclosed
EP-0154245-A2 Process for the fabrication of copolyamides from adipic acid, terephthalic acid and hexamethylene diamine BAYER AG (DE) 1985-09-11 EP disclosed