SCHEMBL8931667

SCHEMBL8931667

CCC(C(=O)c1ccc(Cl)cc1)n1ncn(-c2ccc(N3CCN(c4ccccc4OC)CC3)nc2)c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 3/20 0.47
DRD2 P14416 3/20 0.43
DRD3 P35462 3/20 0.43
DRD4 P21917 2/20 0.43
LMNA P02545 5/20 0.42
MAPK1 P28482 1/20 0.42
MAPT P10636 3/20 0.41
TP53 P04637 1/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 3/20 0.39
HDAC6 Q9UBN7 1/20 0.39
KDM4E B2RXH2 2/20 0.39
GAA P10253 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
TACR2 P21452 1/20 0.39
TACR1 P25103 1/20 0.39
TACR3 P29371 1/20 0.39
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8931761 0.91 DGAT1 (0.54) DGAT1DRD2DRD3DRD4LMNA
SCHEMBL8931751 0.90 DGAT1 (0.49) DGAT1LMNAMAPTNPC1ALDH1A1
SCHEMBL8931744 0.88 DGAT1 (0.48) DGAT1LMNAMAPTALDH1A1KDM4E
SCHEMBL8931682 0.88 DGAT1 (0.48) DGAT1DRD4LMNAMAPTALDH1A1
Hydrochloric Acid SCHEMBL8931688 0.88 DGAT1 (0.47) DGAT1LMNAMAPTALDH1A1KDM4E
SCHEMBL8931730 0.87 MAPT (0.54) DGAT1LMNAMAPK1MAPTTP53
SCHEMBL8814915 0.87 DGAT1 (0.51) DGAT1DRD2DRD4LMNAMAPT
SCHEMBL8927422 0.87 DGAT1 (0.47) DGAT1DRD4LMNAMAPK1MAPT
SCHEMBL8931650 0.86 DGAT1 (0.51) DGAT1DRD2DRD4MAPK1MAPT
SCHEMBL8927419 0.86 DGAT1 (0.47) DGAT1DRD4LMNAMAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5650411-A BACTERICIDES FOR HELICOBACTER DISEASES AND BACTERIA RESISTANCE JANSSEN PHARMACEUTICA N.V. (BE) 1997-07-22 US disclosed
EP-0684821-A1 SUBSTITUTED AZOLONE DERIVATIVES FOR TREATING DISEASES CAUSED BY HELICOBACTER JANSSEN PHARMACEUTICA N.V. (BE) 1995-12-06 EP disclosed
WO-1994018978-A1 SUBSTITUTED AZOLONE DERIVATIVES FOR TREATING DISEASES CAUSED BY HELICOBACTER JANSSEN PHARMACEUTICA N.V. (BE) 1994-09-01 WO disclosed