SCHEMBL8932001

SCHEMBL8932001

CC(CC(CCC(C(=O)O)n1cnc2ccccc21)c1ccccc1-c1nn[nH]n1)C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DNMT3A Q9Y6K1 1/20 0.35
AGTR1 P30556 4/20 0.35
AGTR2 P50052 3/20 0.35
HDAC8 Q9BY41 1/20 0.35
PTPRC P08575 1/20 0.34
PTPN2 P17706 1/20 0.34
PTPN1 P18031 1/20 0.34
APAF1 O14727 1/20 0.34
PDE3A Q14432 3/20 0.33
PDE4A P27815 2/20 0.33
PDE4B Q07343 2/20 0.33
PDE4C Q08493 2/20 0.33
PDE4D Q08499 2/20 0.33
PDE3B Q13370 2/20 0.33
ABCB11 O95342 1/20 0.33
EGFR P00533 1/20 0.33
ERBB2 P04626 1/20 0.33
CYP3A4 P08684 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7015525 0.79 AGTR1 (0.41) AGTR1AGTR2PTPRCPTPN2PTPN1
SCHEMBL7015176 0.70 AGTR1 (0.49) AGTR1AGTR2ABCB11LTB4R2
SCHEMBL7017110 0.70 AGTR1 (0.48) AGTR1AGTR2ABCB11LTB4R2
SCHEMBL7015549 0.69 AGTR1 (0.47) AGTR1AGTR2ABCB11LTB4R2
SCHEMBL8911545 0.68 AGTR1 (0.41) AGTR1AGTR2PDE3AABCB11EGFR
SCHEMBL8931859 0.68 EGLN3 (0.43) APAF1CYP3A4CYP2C9
SCHEMBL3795625 0.67 HDAC8 (0.55) DNMT3AHDAC8APAF1CYP3A4CYP2C9
SCHEMBL8932004 0.66 AGTR1 (0.42) AGTR1AGTR2ABCB11LTB4R2
SCHEMBL7016171 0.65
SCHEMBL8931908 0.65 AGTR1 (0.39) AGTR1AGTR2PDE3AABCB11EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5693633-A Angiotensin II antagonists ELI LILLY AND COMPANY (US) 1997-12-02 US disclosed