SCHEMBL8932026

SCHEMBL8932026

C[N+]1(c2nc3cc(-c4ccccc4C#N)ccc3[nH]2)CCC[C@H]1C(=O)OCc1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OXTR P30559 1/20 0.37
AVPR1A P37288 1/20 0.37
TRPA1 O75762 1/20 0.35
FFAR1 O14842 3/20 0.35
AKR1B1 P15121 1/20 0.35
ABL1 P00519 1/20 0.35
USP30 Q70CQ3 1/20 0.34
TSHR P16473 1/20 0.34
EGLN1 Q9GZT9 2/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PIK3CA P42336 1/20 0.33
MTOR P42345 1/20 0.33
GRIN2B Q13224 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8913033 0.75 GRIN2B (0.42) OXTRAVPR1AUSP30GRIN2B
SCHEMBL7019918 0.66 GAA (0.54) TRPA1TSHRKDM4EALDH1A1GAA
SCHEMBL7015221 0.64 TRPA1 (0.57) TRPA1TSHRKDM4EALDH1A1MAPT
SCHEMBL7020356 0.64 MAPT (0.47) TRPA1KDM4EALDH1A1MAPTHPGD
SCHEMBL2770633 0.62 CYP3A4 (0.58) TRPA1ABL1USP30KDM4EALDH1A1
SCHEMBL3751793 0.62 CYP3A4 (0.58) TRPA1ABL1USP30KDM4EALDH1A1
SCHEMBL9025920 0.62 FFAR1 (0.57) OXTRAVPR1AFFAR1AKR1B1EGLN1
SCHEMBL7014174 0.62 TRPA1 (0.53) TRPA1TSHRKDM4EALDH1A1MAPT
SCHEMBL7014933 0.62 TRPA1 (0.53) TRPA1TSHRKDM4EALDH1A1MAPT
SCHEMBL7019183 0.61 CYP1A2 (0.53) TRPA1TSHRKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5693633-A Angiotensin II antagonists ELI LILLY AND COMPANY (US) 1997-12-02 US disclosed