SCHEMBL8932650

SCHEMBL8932650

COc1ccc2c(c1)c(CC(=O)N1CCOCC1)c(C)n2C(=O)c1ccccc1Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 15/20 1.00
CNR1 P21554 13/20 1.00
TSHR P16473 3/20 0.75
CYP3A4 P08684 2/20 0.75
CYP1A2 P05177 2/20 0.75
CYP2C9 P11712 2/20 0.75
NFKB1 P19838 2/20 0.75
MEN1 O00255 1/20 0.75
GMNN O75496 1/20 0.75
PKM P14618 1/20 0.75
CYP2C19 P33261 1/20 0.75
BLM P54132 1/20 0.75
PMP22 Q01453 1/20 0.75
KMT2A Q03164 1/20 0.75
TP53 P04637 1/20 0.65
HPGD P15428 1/20 0.65
ALOX15 P16050 1/20 0.65
MTOR P42345 1/20 0.65
SMN1; SMN2 Q16637 1/20 0.65
TDP1 Q9NUW8 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8932634 0.87 CNR2 (0.88) CNR2CNR1TSHRCYP3A4CYP1A2
SCHEMBL9089051 0.86 CNR2 (0.87) CNR2CNR1TSHRCYP3A4TP53
Indomethacin Morpholinylamide SCHEMBL8314320 0.85 CNR2 (1.00) CNR2CNR1TSHRCYP3A4CYP1A2
Indomethacin Morpholinylamide SCHEMBL29358919 0.85 CNR2 (1.00) CNR2CNR1TSHRCYP3A4CYP1A2
SCHEMBL6753402 0.84 CNR1 (0.83) CNR2CNR1TSHRCYP1A2CYP2C9
SCHEMBL16870401 0.83 CNR2 (0.86) CNR2CNR1TSHRCYP3A4CYP1A2
SCHEMBL4322359 0.81 CNR2 (0.85) CNR2CNR1TSHRCYP1A2CYP2C9
SCHEMBL8932661 0.81 CNR2 (1.00) CNR2CNR1TSHRCYP3A4CYP1A2
SCHEMBL29835924 0.79 CNR2 (1.00) CNR2CNR1TSHRCYP3A4TP53
SCHEMBL29448220 0.79 CNR2 (1.00) CNR2CNR1TSHRCYP3A4TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996025397-A1 INDOLE DERIVATIVES WITH AFFINITY FOR THE CANNABINOID RECEPTOR MERCK FROSST CANADA INC. (CA) 1996-08-22 WO claimed
WO-1996025397-A1 INDOLE DERIVATIVES WITH AFFINITY FOR THE CANNABINOID RECEPTOR MERCK FROSST CANADA INC. (CA) 1996-08-22 WO disclosed
US-5532237-A INTRAOCULAR FOR TREATMENT OF GLAUCOMA MERCK FROSST CANADA, INC. (CA) 1996-07-02 US disclosed