SCHEMBL8932689

SCHEMBL8932689

Cc1c(CC(=O)O)c2ccccc2n1C(=O)c1cccc2ccccc12

nearest known ligand 0.64

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 7/20 0.64
CNR1 P21554 4/20 0.64
ABCB1 P08183 1/20 0.62
PTGS1 P23219 1/20 0.62
PTGS2 P35354 1/20 0.62
PTGIR P43119 6/20 0.53
LMNA P02545 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
TSHR P16473 1/20 0.50
NFKB1 P19838 1/20 0.50
HIF1A Q16665 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
PTGDR2 Q9Y5Y4 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13802412 0.87 ABCB1 (0.65) CNR2CNR1ABCB1PTGS1PTGS2
SCHEMBL13802382 0.82 ABCB1 (0.60) CNR2CNR1ABCB1PTGS1PTGS2
Delmetacin SCHEMBL286727 0.82 ABCB1 (0.82) ABCB1PTGS1PTGS2PTGIRLMNA
SCHEMBL13802418 0.81 RORC (0.64) CNR2CNR1ABCB1PTGS1PTGS2
SCHEMBL13802389 0.80 ABCB1 (0.70) CNR2CNR1ABCB1PTGS1PTGS2
SCHEMBL13802409 0.79 ABCB1 (0.81) ABCB1PTGS1PTGS2PTGIRLMNA
SCHEMBL13802410 0.79 ABCB1 (0.68) ABCB1PTGS1PTGS2PTGIRLMNA
SCHEMBL4209798 0.78 ABCB1 (0.71) CNR2CNR1ABCB1PTGS1PTGS2
SCHEMBL2982593 0.78 ABCB1 (0.55) CNR2CNR1ABCB1PTGS1PTGS2
SCHEMBL12480026 0.78 ABCB1 (0.64) ABCB1PTGS1PTGS2PTGIRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996025397-A1 INDOLE DERIVATIVES WITH AFFINITY FOR THE CANNABINOID RECEPTOR MERCK FROSST CANADA INC. (CA) 1996-08-22 WO claimed
WO-1996025397-A1 INDOLE DERIVATIVES WITH AFFINITY FOR THE CANNABINOID RECEPTOR MERCK FROSST CANADA INC. (CA) 1996-08-22 WO disclosed
US-5532237-A INTRAOCULAR FOR TREATMENT OF GLAUCOMA MERCK FROSST CANADA, INC. (CA) 1996-07-02 US disclosed