SCHEMBL8932710

SCHEMBL8932710

Cc1oc(-c2ccccc2)nc1Cc1cc2cc(CO)ccc2n1S(=O)(=O)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.46
PPARG P37231 13/20 0.43
PPARA Q07869 11/20 0.43
KDM4E B2RXH2 1/20 0.42
POLB P06746 3/20 0.42
LMNA P02545 1/20 0.42
PPARD Q03181 2/20 0.41
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8932721 0.85 PPARA (0.40) KDRPPARGPPARAKDM4EPOLB
SCHEMBL8932709 0.77 KDR (0.40) KDRPPARGPPARAKDM4EPOLB
SCHEMBL6117631 0.73 CA12 (0.54) PPARGPPARAPPARD
SCHEMBL18416801 0.70 PPARG (0.70) PPARGPPARAPPARD
SCHEMBL7559600 0.68 KDR (0.83) KDRPPARGPPARAMAPT
SCHEMBL4037331 0.68 KDM4E (0.69) KDRPPARGPPARAKDM4ELMNA
SCHEMBL4031706 0.67 KDR (0.57) KDRPPARGPPARAKDM4EPPARD
SCHEMBL6220972 0.67 KDM4E (0.54) PPARGPPARAKDM4ELMNAPPARD
SCHEMBL6860260 0.67 HTR6 (0.59) PPARGPPARAPOLBPPARD
SCHEMBL2928321 0.67 PPARG (0.46) PPARGPPARAKDM4EPOLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996026207-A1 THIAZOLIDINE AND OXAZOLIDINE INDOLES WITH HYPOCLYCEMIC ACTIVITY NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 1996-08-29 WO disclosed