SCHEMBL8933916

SCHEMBL8933916

COc1ccc2c(c1F)CSc1c(C(F)(F)F)nn(-c3ccc(S(C)(=O)=O)cc3)c1-2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 19/20 1.00
PTGS1 P23219 9/20 0.60
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
GRIA2 P42262 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30424119 0.91 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL860766 0.91 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL8934224 0.91 PTGS2 (0.84) PTGS2PTGS1CYP1A2CYP2D6GRIA2
SCHEMBL5071832 0.87 PTGS2 (0.77) PTGS2PTGS1
SCHEMBL13776402 0.87 PTGS2 (0.77) PTGS2PTGS1
SCHEMBL8934166 0.83 PTGS2 (0.84) PTGS2PTGS1
SCHEMBL8937611 0.83 PTGS2 (0.71) PTGS2PTGS1
SCHEMBL8933879 0.82 PTGS2 (0.82) PTGS2PTGS1
SCHEMBL5698663 0.80 PTGS2 (0.82) PTGS2PTGS1CYP1A2CYP2D6GRIA2
SCHEMBL8933882 0.79 PTGS2 (1.00) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996009304-A1 BENZOPYRANOPYRAZOLYL DERIVATIVES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-03-28 WO claimed
US-5565482-A ANTIINFLAMMATORY AGENTS, ANTIARTHRITIC AGENTS G.D. SEARLE & CO. (US) 1996-10-15 US disclosed
US-5547975-A ANTIARTHRIC AGENTS, ANALGESICS AND ANTIPYRETICS; INHIBITORS OF CYCLOOXYGENASE II; SIDE EFFECT REDUCTION G.D. SEARLE & CO. 1996-08-20 US disclosed
WO-1996009304-A1 BENZOPYRANOPYRAZOLYL DERIVATIVES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-03-28 WO disclosed