SCHEMBL8934569

SCHEMBL8934569

CC(=O)CCCc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.58
KCNH2 Q12809 3/20 0.51
KCNJ1 P48048 2/20 0.50
MAPK1 P28482 1/20 0.50
ALDH1A1 P00352 4/20 0.48
MAPT P10636 2/20 0.48
CYP2C19 P33261 2/20 0.48
KMT2A Q03164 2/20 0.48
HTT P42858 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
LOXL2 Q9Y4K0 1/20 0.47
MAOB P27338 1/20 0.47
SIGMAR1 Q99720 1/20 0.46
MEN1 O00255 1/20 0.46
HRH3 Q9Y5N1 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8855273 0.89 TSHR (0.61) TSHRKCNH2KCNJ1MAPK1ALDH1A1
SCHEMBL135651 0.84 TSHR (0.59) TSHRKCNH2KCNJ1MAPK1ALDH1A1
SCHEMBL2850348 0.84 TSHR (0.59) TSHRKCNH2KCNJ1ALDH1A1MAPT
SCHEMBL29465190 0.83 PKM (0.43) TSHRMAPK1ALDH1A1MAPTKMT2A
SCHEMBL8813056 0.83 TSHR (0.58) TSHRKCNH2KCNJ1ALDH1A1MAPT
SCHEMBL7733298 0.83 TSHR (0.58) TSHRKCNH2KCNJ1ALDH1A1MAPT
Hydrochloric Acid SCHEMBL5030930 0.83 TSHR (0.58) TSHRKCNH2KCNJ1MAPK1ALDH1A1
SCHEMBL5030925 0.83 TSHR (0.58) TSHRKCNH2KCNJ1ALDH1A1MAPT
SCHEMBL9763373 0.82 TSHR (0.46) TSHRKCNH2MAPK1ALDH1A1MAPT
SCHEMBL29318769 0.82 TSHR (0.53) TSHRKCNH2KCNJ1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996030350-A1 AMIDINE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-10-03 WO disclosed
EP-0178874-B1 ALKYLSULFONAMIDOPHENYLALKYLAMINES ELI LILLY AND COMPANY (US) 1989-04-05 EP disclosed
US-4596827-A Antiarrhythmia agents ELI LILLY AND COMPANY (US) 1986-06-24 US disclosed
EP-0178874-A1 Alkylsulfonamidophenylalkylamines ELI LILLY AND COMPANY (US) 1986-04-23 EP disclosed
US-4569801-A ANTIARRHYTHMIA AGENTS ELI LILLY AND COMPANY (US) 1986-02-11 US disclosed