Spiperone

Spiperone

SCHEMBL8935119

NC(=S)S.O=C(CCCN1CCC2(CC1)C(=O)NCN2c1ccccc1)c1ccc(F)cc1

nearest known ligand 0.88

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.88
HTR2A P28223 4/20 0.88
DRD3 P35462 4/20 0.88
HTR7 P34969 3/20 0.88
DRD4 P21917 3/20 0.88
CYP1A2 P05177 3/20 0.88
ADRB1 P08588 3/20 0.88
CYP2D6 P10635 3/20 0.88
ADRA2B P18089 3/20 0.88
ADRA2C P18825 3/20 0.88
SLC6A4 P31645 3/20 0.88
ADRA1A P35348 3/20 0.88
HRH1 P35367 3/20 0.88
OPRM1 P35372 3/20 0.88
HTR2B P41595 3/20 0.88
HTR6 P50406 3/20 0.88
SLC6A3 Q01959 3/20 0.88
NPC1 O15118 2/20 0.88
USP2 O75604 2/20 0.88
LMNA P02545 2/20 0.88

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Spiperone SCHEMBL116031 0.94 DRD2 (1.00) DRD2HTR2ADRD3HTR7DRD4
Spiperone SCHEMBL466892 0.93 HTR7 (1.00) DRD2HTR2ADRD3HTR7DRD4
Spiperone SCHEMBL9213600 0.90 DRD2 (0.93) DRD2HTR2ADRD3HTR7DRD4
Fluspiperone SCHEMBL121266 0.89 DRD2 (0.90) DRD2HTR2ADRD3HTR7DRD4
Spiperone SCHEMBL4279344 0.89 DRD2 (0.89) DRD2HTR2ADRD3HTR7DRD4
SCHEMBL10735272 0.87 DRD2 (0.86) DRD2HTR2ADRD3HTR7DRD4
SCHEMBL10729769 0.84 DRD2 (0.82) DRD2HTR2ADRD3HTR7DRD4
SCHEMBL12188097 0.83 DRD2 (0.80) DRD2HTR2ADRD3HTR7DRD4
Spiperone SCHEMBL6160476 0.83 HTR7 (0.81) DRD2HTR2ADRD3HTR7DRD4
Spiperone SCHEMBL10971898 0.83 DRD2 (0.76) DRD2HTR2ADRD3HTR7DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996030054-A1 99mTc - LABELLED SEROTONIN RECEPTOR BINDING SUBSTANCES MALLINCKRODT MEDICAL, INC. (US) 1996-10-03 WO disclosed