SCHEMBL8936088

SCHEMBL8936088

CCOP(=O)(Cc1cc(=O)[nH]c2cc(Cl)cc(Cl)c12)OCC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.36
CA9 Q16790 1/20 0.36
GRIN2D O15399 2/20 0.35
GRIN3B O60391 2/20 0.35
GRIN1 Q05586 2/20 0.35
GRIN2A Q12879 2/20 0.35
GRIN2B Q13224 2/20 0.35
GRIN2C Q14957 2/20 0.35
GRIN3A Q8TCU5 2/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
HPGD P15428 1/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
CYP2C19 P33261 1/20 0.35
BLM P54132 1/20 0.35
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8936210 0.80 GRIN2D (0.54) CA12CA9GRIN2DGRIN3BGRIN1
SCHEMBL8936102 0.79 GRIN2D (0.36) CA12CA9GRIN2DGRIN3BGRIN1
SCHEMBL8936157 0.73 CA12 (0.44) CA12CA9GRIN2DGRIN3BGRIN1
SCHEMBL8936172 0.72 SMN1; SMN2 (0.49) CA9GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL10627650 0.70 TDP1 (0.46) MEN1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL8936072 0.69 SMN1; SMN2 (0.38) MEN1HPGDALOX15KMT2A
SCHEMBL15316683 0.67 TDP1 (0.43) MEN1HPGDTSHRKMT2ATDP1
SCHEMBL6298909 0.67 TSHR (0.46) MEN1TSHRKMT2ATDP1
SCHEMBL901666 0.67 HSD17B10 (0.41) TSHR
SCHEMBL23908226 0.66 TSHR (0.50) MEN1TSHRKMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510338-A ADMINISTERING TO A MAMMAL TO RELIEVE PAIN AND TO TREAT CONVULSIONS, CEREBRAL ISCHEMIC DAMAGE, AND EMESIS GUILFORD PHARMACEUTICALS INC. (US) 1996-04-23 US disclosed
US-5342946-A Phosphonoalkylquinolin-2-ones as novel antagonists of non-NMDA ionotropic excitatory amino acid receptors GUILFORD PHARMACEUTICALS INC. (US) 1994-08-30 US disclosed