SCHEMBL8936319

SCHEMBL8936319

O=C1C=CC=c2cc3c(cc21)=Cc1ccccc1CC3

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 1/20 0.33
CES1 P23141 1/20 0.33
NISCH Q9Y2I1 1/20 0.32
KDM1A O60341 1/20 0.32
PTGS2 P35354 1/20 0.30
HTR1A P08908 1/20 0.30
DRD2 P14416 1/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
HTR7 P34969 1/20 0.30
HRH1 P35367 1/20 0.30
DRD3 P35462 1/20 0.30
HTR2B P41595 1/20 0.30
CYP19A1 P11511 1/20 0.30
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL440760 0.77 CDC25B (0.38) CES1
SCHEMBL2452850 0.75 IDO1 (0.41) CES1
SCHEMBL126239 0.72 CDC25B (0.33)
SCHEMBL26205058 0.69 NQO1 (0.31)
SCHEMBL11311853 0.67 CDC25B (0.31)
SCHEMBL8321788 0.65
SCHEMBL10533241 0.65
SCHEMBL10537369 0.64
SCHEMBL20511815 0.63 PARP1 (0.46) GPR84CES1NISCHKDM1AHTR1A
SCHEMBL20511816 0.63 PARP1 (0.46) GPR84CES1NISCHKDM1AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996031469-A1 N-SUBSTITUTED AZAHETEROCYCLIC CARBOXYLIC ACIDS AND ESTERS THEREOF NOVO NORDISK A/S (DK) 1996-10-10 WO disclosed