SCHEMBL8936565

SCHEMBL8936565

Cc1cc2c(-c3c(C)cccc3C)c(NC(=O)NCc3ccccc3Cl)n(C)c(=O)c2cc1C

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 9/20 0.61
NPC1 O15118 3/20 0.45
RAB9A P51151 2/20 0.45
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
PTGER3 P43115 1/20 0.41
LMNA P02545 1/20 0.41
ALDH1A1 P00352 1/20 0.41
TP53 P04637 1/20 0.41
THRB P10828 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8936447 0.92 TACR1 (0.53) TACR1NPC1RAB9AMEN1KMT2A
SCHEMBL8936575 0.91 TACR1 (0.60) TACR1NPC1RAB9AMEN1KMT2A
SCHEMBL8936460 0.90 TACR1 (0.76) TACR1NPC1RAB9AMEN1KMT2A
SCHEMBL8936514 0.88 TACR1 (0.59) TACR1NPC1RAB9AMEN1KMT2A
SCHEMBL8936431 0.83 TACR1 (0.56) TACR1NPC1RAB9AMEN1KMT2A
SCHEMBL8936536 0.83 TACR1 (0.77) TACR1NPC1RAB9A
SCHEMBL8936580 0.82 TACR1 (0.80) TACR1NPC1RAB9AMEN1KMT2A
SCHEMBL8936410 0.82 TACR1 (0.72) TACR1NPC1RAB9AALDH1A1
SCHEMBL8936599 0.80 TACR1 (0.76) TACR1NPC1RAB9AALDH1A1
SCHEMBL8936556 0.78 TACR1 (0.53) TACR1NPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5523305-A ANALGESICS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-06-04 US disclosed
EP-0566069-A1 Tachykinin receptor antagonists, isoquinolones and their production TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-10-20 EP disclosed