SCHEMBL8936623

SCHEMBL8936623

CCN1C(=O)c2cccc(C)c2Oc2ncccc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.45
ALDH1A1 P00352 4/20 0.45
CASP1 P29466 3/20 0.45
PKM P14618 2/20 0.45
CASP7 P55210 2/20 0.45
ALOX15 P16050 1/20 0.45
MAPK1 P28482 1/20 0.45
HPGD P15428 1/20 0.45
MPI P34949 1/20 0.45
CACNA1B Q00975 1/20 0.45
APBA1 Q02410 1/20 0.45
MAPT P10636 7/20 0.41
LMNA P02545 2/20 0.41
BRD4 O60885 1/20 0.40
POLB P06746 2/20 0.39
CYP1B1 Q16678 1/20 0.38
TP53 P04637 1/20 0.38
KDM4E B2RXH2 1/20 0.38
APAF1 O14727 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8936638 0.86 BRD4 (0.44) SMN1; SMN2ALDH1A1CASP1PKMCASP7
SCHEMBL8936588 0.77 MAPT (0.50) SMN1; SMN2MAPTLMNAPOLBGAA
SCHEMBL9101435 0.75 TP53 (0.60) SMN1; SMN2MAPTLMNAPOLBTP53
SCHEMBL9369130 0.74 ALDH1A1 (0.47) SMN1; SMN2ALDH1A1CASP1PKMCASP7
SCHEMBL9368959 0.72 AKT1 (0.47) SMN1; SMN2ALDH1A1CASP1PKMCASP7
SCHEMBL9099840 0.72 MAPT (0.58) SMN1; SMN2MAPTLMNAPOLBGAA
SCHEMBL8301100 0.70 ALDH1A1 (0.50) SMN1; SMN2ALDH1A1CASP1PKMCASP7
SCHEMBL8791051 0.70 BRD4 (0.51) SMN1; SMN2ALDH1A1CASP1PKMCASP7
SCHEMBL9369777 0.69 BRD4 (0.50) SMN1; SMN2ALDH1A1CASP1PKMCASP7
SCHEMBL8301745 0.68 ALDH1A1 (0.54) SMN1; SMN2ALDH1A1CASP1PKMCASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5547951-A ENZYME INHIBITORS; AIDS BOEHRINGER INGELHEIM PHARAMCEUTICALS, INC. (US) 1996-08-20 US disclosed
EP-0417534-A1 Pyrido[2,3-b][1,4]benzoxazepin (and thiazepin)-6(5H)-ones and thiones and their use in the prevention or treatment of AIDS Boehringer Ingelheim Pharmaceuticals Inc. (US) 1991-03-20 EP disclosed