SCHEMBL8936757

SCHEMBL8936757

Oc1ccc(C(F)(F)F)cc1Cn1cncn1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.48
CYP19A1 P11511 11/20 0.44
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ALOX15 P16050 1/20 0.43
KMT2A Q03164 1/20 0.39
HSP90AA1 P07900 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
LRRK2 Q5S007 1/20 0.38
UGT1A4 P22310 1/20 0.38
PDE4D Q08499 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9202210 0.81 BRD4 (0.51) BRD4CYP19A1CYP3A4CYP2C9CYP2C19
SCHEMBL9198430 0.81 BRD4 (0.46) BRD4CYP19A1CYP1A2CYP3A4CYP2C9
SCHEMBL8936696 0.78 BRD4 (0.51) BRD4CYP19A1CYP1A2CYP3A4CYP2C9
SCHEMBL8936736 0.78 CYP19A1 (0.53) BRD4CYP19A1CYP3A4CYP2C9CYP2C19
SCHEMBL9202769 0.78 BRD4 (0.51) BRD4CYP19A1HDAC1HDAC6
SCHEMBL9197402 0.74 CYP19A1 (0.56) BRD4CYP19A1KMT2A
SCHEMBL8507241 0.74 CYP19A1 (0.60) CYP19A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8936807 0.73 CYP19A1 (0.58) BRD4CYP19A1CYP2C19KDM4EHSP90AA1
SCHEMBL14476866 0.72 CYP19A1 (0.56) CYP19A1HDAC1HDAC6UGT1A4PDE4D
SCHEMBL9826863 0.70 HSP90AA1 (0.54) CYP19A1CYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587392-A THERAPY FOR ESTROGEN DEPENDENT DISEASES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1996-12-24 US disclosed
EP-0684235-A1 Novel azolyl methyl phenyl derivatives having aromatase inhibitory activity MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1995-11-29 EP disclosed