SCHEMBL8936771

SCHEMBL8936771

CNc1cc(Oc2ccc(Cl)cc2Cn2cncn2)ccc1[N+](=O)[O-]

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.41
PKM P14618 2/20 0.41
CCR1 P32246 1/20 0.41
CCR2 P41597 1/20 0.41
CCR4 P51679 1/20 0.41
SCN9A Q15858 1/20 0.38
PDE7A Q13946 1/20 0.38
HTR2A P28223 3/20 0.38
SLC6A4 P31645 3/20 0.38
KCNH2 Q12809 3/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
POLB P06746 1/20 0.36
CYP19A1 P11511 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9201309 0.93 CCR1 (0.45) TDP1PKMCCR1CCR2CCR4
SCHEMBL8936766 0.91 MAPT (0.41) TDP1PKMCCR1CCR2CCR4
SCHEMBL9196269 0.90 CYP19A1 (0.43) PKMSCN9AHTR2ASLC6A4MAPT
SCHEMBL8936755 0.89 PKM (0.41) TDP1PKMSCN9AHTR2ASLC6A4
SCHEMBL9201983 0.89 PKM (0.41) TDP1PKMCCR1CCR2CCR4
SCHEMBL9198771 0.89 PKM (0.41) PKMSCN9AHTR2ASLC6A4KCNH2
SCHEMBL8936748 0.88 PKM (0.41) PKMSCN9AHTR2ASLC6A4KCNH2
SCHEMBL9202877 0.87 PKM (0.40) PKMSCN9ASLC6A4CYP19A1
SCHEMBL8936739 0.86 MEN1 (0.40) TDP1PKMHTR2ASLC6A4KCNH2
SCHEMBL8936735 0.86 PDE7A (0.45) TDP1PKMCCR1CCR2CCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587392-A THERAPY FOR ESTROGEN DEPENDENT DISEASES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1996-12-24 US disclosed
EP-0684235-A1 Novel azolyl methyl phenyl derivatives having aromatase inhibitory activity MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1995-11-29 EP disclosed